Search Count: 69
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Crystal Structure Of Kras G12D In Complex With Gdp And Compound 5
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.35 Å Release Date: 2023-11-08 Classification: ONCOPROTEIN/INHIBITOR Ligands: GDP, MG, VM9 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-11-08
Ligands: GDP, MG, VM9
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Crystal Structure Of Kras G12D In Complex With Gdp And Compound 8
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.50 Å Release Date: 2023-11-08 Classification: ONCOPROTEIN/INHIBITOR Ligands: GDP, MG, VQT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-11-08
Ligands: GDP, MG, VQT
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Crystal Structure Of Kras G12D In Complex With Gdp And Compound 14
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.20 Å Release Date: 2023-11-08 Classification: ONCOPROTEIN/INHIBITOR Ligands: GDP, MG, VR5 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-11-08
Ligands: GDP, MG, VR5
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Voltage-Gated Potassium Channel Kv3.1 With Novel Positive Modulator (9M)-9-{5-Chloro-6-[(3,3-Dimethyl-2,3-Dihydro-1-Benzofuran-4-Yl)Oxy]-4-Methylpyridin-3-Yl}-2-Methyl-7,9-Dihydro-8H-Purin-8-One (Compound 4)
Organism: Homo sapiens
Method: ELECTRON MICROSCOPY Release Date: 2023-10-25 Classification: TRANSPORT PROTEIN Ligands: ZN, X9T, POV, K |
Organism: Homo sapiens
Method: ELECTRON MICROSCOPY
Release Date: 2023-10-25
Ligands: ZN, X9T, POV, K
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Voltage-Gated Potassium Channel Kv3.1 Apo
Organism: Homo sapiens
Method: ELECTRON MICROSCOPY Release Date: 2023-10-25 Classification: TRANSPORT PROTEIN Ligands: ZN, CLR, K |
Organism: Homo sapiens
Method: ELECTRON MICROSCOPY
Release Date: 2023-10-25
Ligands: ZN, CLR, K
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Prmt5:Mep50 Complexed With Inhibitor Pf-06939999
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.49 Å Release Date: 2021-11-17 Classification: TRANSFERASE/Transcription Ligands: ZR1 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-11-17
Ligands: ZR1
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Prmt5:Mep50 Complexed With Inhibitor Pf-06855800
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.71 Å Release Date: 2021-11-17 Classification: Transferase/Transcription Ligands: ZR4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-11-17
Ligands: ZR4
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Prmt5:Mep50 Complexed With Adenosine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.41 Å Release Date: 2021-11-17 Classification: TRANSFERASE/Transcription Ligands: ADN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-11-17
Ligands: ADN
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Prmt5(M420T Mutant):Mep50 Complexed With Inhibitor Pf-06855800
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2021-11-17 Classification: TRANSFERASE/Transcription Ligands: ZR4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-11-17
Ligands: ZR4
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Prmt5(M420T Mutant):Mep50 Complexed With Inhibitor Pf-06939999
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.55 Å Release Date: 2021-11-17 Classification: transferase/Transcription Ligands: ZR1 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-11-17
Ligands: ZR1
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Crystal Structure Of Mbp-Trem2 Ig Domain Fusion With Fragment, 2-((4-Bromophenyl)Amino)Ethan-1-Ol
Organism: Methanosarcina mazei, Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.47 Å Release Date: 2021-02-17 Classification: SIGNALING PROTEIN Ligands: V5S, DMS |
Organism: Methanosarcina mazei, Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-02-17
Ligands: V5S, DMS
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Orexin Receptor 2 (Ox2R) In Complex With G Protein And Natural Peptide-Agonist Orexin B (Oxb)
Organism: Homo sapiens, Mus musculus
Method: ELECTRON MICROSCOPY Release Date: 2021-02-10 Classification: MEMBRANE PROTEIN |
Organism: Homo sapiens, Mus musculus
Method: ELECTRON MICROSCOPY
Release Date: 2021-02-10
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Orexin Receptor 2 (Ox2R) In Complex With G Protein And Small-Molecule Agonist Compound 1
Organism: Homo sapiens, Mus musculus, Lama glama
Method: ELECTRON MICROSCOPY Release Date: 2021-02-10 Classification: MEMBRANE PROTEIN Ligands: XGD |
Organism: Homo sapiens, Mus musculus, Lama glama
Method: ELECTRON MICROSCOPY
Release Date: 2021-02-10
Ligands: XGD
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Crystal Structure Of Pi3Kalpha Selective Inhibitor Pf-06843195
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.41 Å Release Date: 2021-01-06 Classification: SIGNALING PROTEIN, Transferase Ligands: VXY |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-01-06
Ligands: VXY
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Crystal Structure Of Pi3Kalpha Selective Inhibitor 11-1575
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.77 Å Release Date: 2021-01-06 Classification: SIGNALING PROTEIN, Transferase Ligands: VY4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-01-06
Ligands: VY4
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Crystal Structure Of Pi3Kalpha Inhibitor 10-5429
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.74 Å Release Date: 2021-01-06 Classification: SIGNALING PROTEIN, Transferase Ligands: VY1 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-01-06
Ligands: VY1
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Crystal Structure Of Pi3Kalpha Inhibitor 4-0686
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.90 Å Release Date: 2021-01-06 Classification: SIGNALING PROTEIN, Transferase Ligands: VYP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-01-06
Ligands: VYP
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Structure Of Human Anaplastic Lymphoma Kinase Domain
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2019-02-20 Classification: TRANSFERASE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-02-20
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Structure Of Hs/Acprc2 In Complex With 5,8-Dichloro-2-[(4-Methoxy-6-Methyl-2-Oxo-1,2-Dihydropyridin-3-Yl)Methyl]-7-[(R)-Methoxy(Oxetan-3-Yl)Methyl]-3,4-Dihydroisoquinolin-1(2H)-One
Organism: Anolis carolinensis, Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.81 Å Release Date: 2017-12-27 Classification: Transferase/Transferase Inhibitor Ligands: ZN, CJD |
Organism: Anolis carolinensis, Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-12-27
Ligands: ZN, CJD
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Structure Of Hs/Acprc2 In Complex With 5,8-Dichloro-7-(3,5-Dimethyl-1,2-Oxazol-4-Yl)-2-[(4,6-Dimethyl-2-Oxo-1,2-Dihydropyridin-3-Yl)Methyl]-3,4-Dihydroisoquinolin-1(2H)-One
Organism: Anolis carolinensis, Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.05 Å Release Date: 2017-12-27 Classification: METAL BINDING PROTEIN Ligands: ZN, CJG |
Organism: Anolis carolinensis, Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-12-27
Ligands: ZN, CJG
