Search Count: 26
![]() |
Crystal Structure Of Wild-Type Egfr In Complex With The Reversible Inhibitor Sevabertinib (Bay 2927088)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.14 Å Release Date: 2025-10-15 Classification: TRANSFERASE Ligands: SIN, CL, DMS, EDO, A1JBI |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-10-15
Ligands: SIN, CL, DMS, EDO, A1JBI
![]() |
Crystal Structure Of Human Map4K1 With An Inhibitor, Bay-405
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2024-06-26 Classification: TRANSFERASE Ligands: GOL, XON |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-06-26
Ligands: GOL, XON
![]() |
Crystal Structure Of Map4K1 With A Smol Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.70 Å Release Date: 2024-06-26 Classification: TRANSFERASE Ligands: XOH |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-06-26
Ligands: XOH
![]() |
Crystal Structure Of Map4K1 With A Smol Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2024-06-26 Classification: TRANSFERASE Ligands: XOR |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-06-26
Ligands: XOR
![]() |
Crystal Structure Of Mst1 With A Map4K1 Smol Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2024-06-26 Classification: TRANSFERASE Ligands: XOZ, GOL, CXS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-06-26
Ligands: XOZ, GOL, CXS
![]() |
Crystal Structure Of Mst1 With A Map4K1 Smol Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.14 Å Release Date: 2024-06-26 Classification: TRANSFERASE Ligands: ASP, XQL, GOL, CXS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-06-26
Ligands: ASP, XQL, GOL, CXS
![]() |
Crystal Structure Of Compound 1 With Erk5
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.47 Å Release Date: 2019-02-27 Classification: TRANSFERASE Ligands: G92 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-02-27
Ligands: G92
![]() |
Crystal Structure Of Compound 35 With Erk5
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.33 Å Release Date: 2019-02-27 Classification: TRANSFERASE Ligands: G9E |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-02-27
Ligands: G9E
![]() |
Ras Guanine Nucleotide Exchange Factor Sos1 (Rem-Cdc25) In New Crystal Form
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2019-02-06 Classification: SIGNALING PROTEIN Ligands: EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-02-06
Ligands: EDO
![]() |
Ras Guanine Nucleotide Exchange Factor Sos1 (Rem-Cdc25) In Complex With Small Molecule Inhibitor Compound 1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2019-02-06 Classification: SIGNALING PROTEIN Ligands: EDO, AXE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-02-06
Ligands: EDO, AXE
![]() |
Ras Guanine Nucleotide Exchange Factor Sos1 (Rem-Cdc25) In Complex With Small Molecule Inhibitor Compound 17
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.01 Å Release Date: 2019-02-06 Classification: SIGNALING PROTEIN Ligands: AWT, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-02-06
Ligands: AWT, EDO
![]() |
Ras Guanine Nucleotide Exchange Factor Sos1 (Rem-Cdc25) In Complex With Small Molecule Inhibitor Compound 18
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2019-02-06 Classification: SIGNALING PROTEIN Ligands: AWZ, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-02-06
Ligands: AWZ, EDO
![]() |
Ras Guanine Nucleotide Exchange Factor Sos1 (Rem-Cdc25) In Complex With Small Molecule Inhibitor Compound 21
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2019-02-06 Classification: SIGNALING PROTEIN Ligands: AWW, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-02-06
Ligands: AWW, EDO
![]() |
Ras Guanine Nucleotide Exchange Factor Sos1 (Rem-Cdc25) In Complex With Small Molecule Inhibitor Bay-293 (Compound 23)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2019-02-06 Classification: SIGNALING PROTEIN Ligands: AXH, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-02-06
Ligands: AXH, EDO
![]() |
Ras Guanine Nucleotide Exchange Factor Sos2 (Rem-Cdc25), With Surface Mutations
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.72 Å Release Date: 2019-02-06 Classification: SIGNALING PROTEIN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-02-06
![]() |
Ras Guanine Exchange Factor Sos1 (Rem-Cdc25) In Complex With Kras(G12C)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.55 Å Release Date: 2019-02-06 Classification: SIGNALING PROTEIN Ligands: GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-02-06
Ligands: GOL
![]() |
Ras Guanine Nucleotide Exchange Factor Sos1 (Rem-Cdc25) In Complex With Kras(G12C) And Fragment Screening Hit F1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2019-02-06 Classification: SIGNALING PROTEIN Ligands: GOL, BQ5 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-02-06
Ligands: GOL, BQ5
![]() |
Ras Guanine Exchange Factor Sos1 (Rem-Cdc25) In Complex With Kras(G12C) And Fragment Screening Hit F2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2019-02-06 Classification: SIGNALING PROTEIN Ligands: GOL, BQ2, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-02-06
Ligands: GOL, BQ2, DMS
![]() |
Ras Guanine Exchange Factor Sos1 (Rem-Cdc25) In Complex With Kras(G12C) And Fragment Screening Hit F3
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2019-02-06 Classification: SIGNALING PROTEIN Ligands: GOL, BPW |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-02-06
Ligands: GOL, BPW
![]() |
Ras Guanine Exchange Factor Sos1 (Rem-Cdc25) In Complex With Kras(G12C) And Fragment Screening Hit F4
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2019-02-06 Classification: SIGNALING PROTEIN Ligands: GOL, BOQ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-02-06
Ligands: GOL, BOQ
