Search Count: 22
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Crystal Structure Analysis Of Thrombin In Complex With Compound D58
Organism: Homo sapiens, Hirudo medicinalis
Method: X-RAY DIFFRACTION Resolution:1.61 Å Release Date: 2014-06-11 Classification: hydrolase/hydrolase inhibitor Ligands: NAG, NA, 7R9 |
Organism: Homo sapiens, Hirudo medicinalis
Method: X-RAY DIFFRACTION
Release Date: 2014-06-11
Ligands: NAG, NA, 7R9
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Crystal Structure Analysis Of Thrombin In Complex With Compound D57, 5-Chlorothiophene-2-Carboxylic Acid [(S)-2-[2-Methyl-3-(2- Oxopyrrolidin-1-Yl)Benzenesulfonylamino]-3-(4-Methylpiperazin-1- Yl)-3-Oxopropyl]Amide (Sar107375)
Organism: Homo sapiens, Hirudo medicinalis
Method: X-RAY DIFFRACTION Resolution:1.77 Å Release Date: 2014-06-04 Classification: hydrolase/hydrolase inhibitor Ligands: NAG, NA, 6XS |
Organism: Homo sapiens, Hirudo medicinalis
Method: X-RAY DIFFRACTION
Release Date: 2014-06-04
Ligands: NAG, NA, 6XS
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Factor Xa In Complex With The Dual Thrombin-Fxa Inhibitor 58.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2013-12-25 Classification: HYDROLASE Ligands: CA, 7R9 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-12-25
Ligands: CA, 7R9
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Factor Xa In Complex With The Dual Thrombin-Fxa Inhibitor 31.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.59 Å Release Date: 2013-12-18 Classification: HYDROLASE Ligands: CA, VYR |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-12-18
Ligands: CA, VYR
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Factor Xa In Complex With The Dual Thrombin-Fxa Inhibitor 57.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.37 Å Release Date: 2013-12-18 Classification: HYDROLASE Ligands: CA, 6XS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-12-18
Ligands: CA, 6XS
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Crystal Structure Of Human Prorenin
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.93 Å Release Date: 2012-05-23 Classification: HYDROLASE Ligands: NAG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-05-23
Ligands: NAG
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Structure-Based Optimization Of Potent 4- And 6-Azaindole-3-Carboxamides As Renin Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2011-08-31 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: NAG, GOL, S53 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-08-31
Ligands: NAG, GOL, S53
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Crystal Structure Analysis Of Renin-Indole-Piperazin Inhibitor Complexes
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.55 Å Release Date: 2010-10-27 Classification: HYDROLASE Ligands: NAG, SSR |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-10-27
Ligands: NAG, SSR
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Crystal Structure Analysis Of Renin-Indole-Piperazin Inhibitor Complexes
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.90 Å Release Date: 2010-10-27 Classification: HYDROLASE Ligands: NAG, S52, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-10-27
Ligands: NAG, S52, GOL
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Crystal Structure Analysis Of Renin-Indole-Piperazine Inhibitor Complexes
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.78 Å Release Date: 2010-10-13 Classification: HYDROLASE Ligands: NAG, S51 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-10-13
Ligands: NAG, S51
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Prolyl Oligopeptidase Complexed With R-Pro-(Decarboxy-Pro)-Type Inhibitors
Organism: Sus scrofa
Method: X-RAY DIFFRACTION Resolution:2.89 Å Release Date: 2009-08-25 Classification: HYDROLASE Ligands: X99 |
Organism: Sus scrofa
Method: X-RAY DIFFRACTION
Release Date: 2009-08-25
Ligands: X99
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Prolyl Oligopeptidase Complexed With R-Pro-(Decarboxy-Pro)-Type Inhibitors
Organism: Sus scrofa
Method: X-RAY DIFFRACTION Resolution:2.73 Å Release Date: 2009-08-25 Classification: Hydrolase/Hydrolase inhibitor Ligands: X98 |
Organism: Sus scrofa
Method: X-RAY DIFFRACTION
Release Date: 2009-08-25
Ligands: X98
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Prolyl Oligopeptidase Complexed With R-Pro-(Decarboxy-Pro)-Type Inhibitors
Organism: Sus scrofa
Method: X-RAY DIFFRACTION Resolution:2.47 Å Release Date: 2009-08-25 Classification: Hydrolase/Hydrolase inhibitor Ligands: X97 |
Organism: Sus scrofa
Method: X-RAY DIFFRACTION
Release Date: 2009-08-25
Ligands: X97
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Crystal Structure Analysis Of The Mutant S189D Rat Chymotrypsin
Organism: Rattus norvegicus
Method: X-RAY DIFFRACTION Resolution:2.55 Å Release Date: 2003-06-10 Classification: HYDROLASE Ligands: CA |
Organism: Rattus norvegicus
Method: X-RAY DIFFRACTION
Release Date: 2003-06-10
Ligands: CA
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Calmodulin Complexed With N-(3,3,-Diphenylpropyl)-N'-[1-R-(3,4-Bis-Butoxyphenyl)-Ethyl]-Propylenediamine (Dpd), 1:2 Complex
Organism: Bos taurus
Method: X-RAY DIFFRACTION Resolution:2.64 Å Release Date: 2000-03-28 Classification: CALCIUM-BINDING PROTEIN Ligands: CA, DPD |
Organism: Bos taurus
Method: X-RAY DIFFRACTION
Release Date: 2000-03-28
Ligands: CA, DPD
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Calmodulin Complexed With N-(3,3,-Diphenylpropyl)-N'-[1-R-(3,4-Bis-Butoxyphenyl)-Ethyl]-Propylenediamine (Dpd)
Organism: Bos taurus
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2000-03-28 Classification: CALCIUM-BINDING PROTEIN Ligands: CA, DPD |
Organism: Bos taurus
Method: X-RAY DIFFRACTION
Release Date: 2000-03-28
Ligands: CA, DPD
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Prolyl Oligopeptidase From Porcine Muscle
Organism: Sus scrofa
Method: X-RAY DIFFRACTION Resolution:1.40 Å Release Date: 1999-05-13 Classification: HYDROLASE Ligands: SGL, SGM, GOL |
Organism: Sus scrofa
Method: X-RAY DIFFRACTION
Release Date: 1999-05-13
Ligands: SGL, SGM, GOL
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Prolyl Oligopeptidase From Porcine Muscle With Covalently Bound Inhibitor Z-Pro-Prolinal
Organism: Sus scrofa
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 1999-05-13 Classification: HYDROLASE Ligands: ZPR |
Organism: Sus scrofa
Method: X-RAY DIFFRACTION
Release Date: 1999-05-13
Ligands: ZPR
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Calmodulin Complexed With Trifluoperazine (1:2 Complex)
Organism: Bos taurus
Method: X-RAY DIFFRACTION Resolution:2.74 Å Release Date: 1998-09-16 Classification: CALCIUM-BINDING PROTEIN Ligands: CA, TFP |
Organism: Bos taurus
Method: X-RAY DIFFRACTION
Release Date: 1998-09-16
Ligands: CA, TFP
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D254E, D256E Mutant Of D-Xylose Isomerase Complexed With Al3 And Xylitol
Organism: Arthrobacter sp. nrrl
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 1998-01-28 Classification: ISOMERASE Ligands: XYL, AL |
Organism: Arthrobacter sp. nrrl
Method: X-RAY DIFFRACTION
Release Date: 1998-01-28
Ligands: XYL, AL
