Search Count: 14
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Crystal Structure Of The Mycobacterium Tuberculosis Transcriptional Repressor Ethr2 In Complex With Bdm41420
Organism: Mycobacterium tuberculosis
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2017-04-26 Classification: TRANSCRIPTION Ligands: 69Y |
Organism: Mycobacterium tuberculosis
Method: X-RAY DIFFRACTION
Release Date: 2017-04-26
Ligands: 69Y
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Iodinated Form Of The Mycobacterium Tuberculosis Repressor Ethr2
Organism: Mycobacterium tuberculosis h37rv
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2017-04-26 Classification: DNA BINDING PROTEIN Ligands: IOD |
Organism: Mycobacterium tuberculosis h37rv
Method: X-RAY DIFFRACTION
Release Date: 2017-04-26
Ligands: IOD
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Unliganded Form Of The Mycobacterium Tuberculosis Repressor Ethr2
Organism: Mycobacterium tuberculosis h37rv
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2017-04-26 Classification: DNA BINDING PROTEIN |
Organism: Mycobacterium tuberculosis h37rv
Method: X-RAY DIFFRACTION
Release Date: 2017-04-26
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Rapid And Efficient Design Of New Inhibitors Of Mycobacterium Tuberculosis Transcriptional Repressor Ethr Using Fragment Growing, Merging And Linking Approaches
Organism: Mycobacterium tuberculosis
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2014-06-25 Classification: TRANSCRIPTION REPRESSOR/INHIBITOR Ligands: 2B2 |
Organism: Mycobacterium tuberculosis
Method: X-RAY DIFFRACTION
Release Date: 2014-06-25
Ligands: 2B2
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Rapid And Efficient Design Of New Inhibitors Of Mycobacterium Tuberculosis Transcriptional Repressor Ethr Using Fragment Growing, Merging And Linking Approaches
Organism: Mycobacterium tuberculosis
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2014-06-25 Classification: TRANSCRIPTION REPRESSOR/INHIBITOR Ligands: 2H2 |
Organism: Mycobacterium tuberculosis
Method: X-RAY DIFFRACTION
Release Date: 2014-06-25
Ligands: 2H2
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Rapid And Efficient Design Of New Inhibitors Of Mycobacterium Tuberculosis Transcriptional Repressor Ethr Using Fragment Growing, Merging And Linking Approaches
Organism: Mycobacterium tuberculosis
Method: X-RAY DIFFRACTION Resolution:2.11 Å Release Date: 2014-06-25 Classification: TRANSCRIPTION REPRESSOR/INHIBITOR Ligands: 2B3 |
Organism: Mycobacterium tuberculosis
Method: X-RAY DIFFRACTION
Release Date: 2014-06-25
Ligands: 2B3
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Rapid And Efficient Design Of New Inhibitors Of Mycobacterium Tuberculosis Transcriptional Repressor Ethr Using Fragment Growing, Merging And Linking Approaches
Organism: Mycobacterium tuberculosis
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2014-06-25 Classification: TRANSCRIPTION REPRESSOR/INHIBITOR Ligands: 2D1 |
Organism: Mycobacterium tuberculosis
Method: X-RAY DIFFRACTION
Release Date: 2014-06-25
Ligands: 2D1
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Rapid And Efficient Design Of New Inhibitors Of Mycobacterium Tuberculosis Transcriptional Repressor Ethr Using Fragment Growing, Merging And Linking Approaches
Organism: Mycobacterium tuberculosis
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2014-06-25 Classification: TRANSCRIPTION REPRESSOR/INHIBITOR Ligands: 2G1 |
Organism: Mycobacterium tuberculosis
Method: X-RAY DIFFRACTION
Release Date: 2014-06-25
Ligands: 2G1
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G106W Mutant Of Ethr From Mycobacterium Tuberculosis
Organism: Mycobacterium tuberculosis
Method: X-RAY DIFFRACTION Resolution:3.20 Å Release Date: 2011-12-28 Classification: TRANSCRIPTION |
Organism: Mycobacterium tuberculosis
Method: X-RAY DIFFRACTION
Release Date: 2011-12-28
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Ethr From Mycobacterium Tuberculosis In Complex With Compound Bdm33066
Organism: Mycobacterium tuberculosis
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2011-12-21 Classification: TRANSCRIPTION/TRANSCRIPTION INHIBITOR Ligands: LL5, GOL |
Organism: Mycobacterium tuberculosis
Method: X-RAY DIFFRACTION
Release Date: 2011-12-21
Ligands: LL5, GOL
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Structural Activation Of The Transcriptional Repressor Ethr From M. Tuberculosis By Single Amino-Acid Change Mimicking Natural And Synthetic Ligands
Organism: Mycobacterium tuberculosis
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2011-12-21 Classification: TRANSCRIPTION/INHIBITOR Ligands: FO5 |
Organism: Mycobacterium tuberculosis
Method: X-RAY DIFFRACTION
Release Date: 2011-12-21
Ligands: FO5
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Structure Of Hth-Type Transcriptional Regulator Ethr, G106W Mutant
Organism: Mycobacterium tuberculosis
Method: X-RAY DIFFRACTION Resolution:1.86 Å Release Date: 2011-12-21 Classification: TRANSCRIPTION |
Organism: Mycobacterium tuberculosis
Method: X-RAY DIFFRACTION
Release Date: 2011-12-21
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Ethionamide Boosters Part 2: Combining Bioisosteric Replacement And Structure-Based Drug Design To Solve Pharmacokinetic Issues In A Series Of Potent 1,2,4-Oxadiazole Ethr Inhibitors.
Organism: Mycobacterium tuberculosis
Method: X-RAY DIFFRACTION Resolution:1.87 Å Release Date: 2011-12-07 Classification: TRANSCRIPTION REPRESSOR/INHIBITOR Ligands: 3SE |
Organism: Mycobacterium tuberculosis
Method: X-RAY DIFFRACTION
Release Date: 2011-12-07
Ligands: 3SE
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Ethionamide Boosters Part 2: Combining Bioisosteric Replacement And Structure-Based Drug Design To Solve Pharmacokinetic Issues In A Series Of Potent 1,2,4-Oxadiazole Ethr Inhibitors.
Organism: Mycobacterium tuberculosis
Method: X-RAY DIFFRACTION Resolution:2.31 Å Release Date: 2011-12-07 Classification: TRANSCRIPTION REPRESSOR/INHIBITOR Ligands: 3SF |
Organism: Mycobacterium tuberculosis
Method: X-RAY DIFFRACTION
Release Date: 2011-12-07
Ligands: 3SF
