Search Count: 16
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Eed In Complex With Prc2 Allosteric Inhibitor Compound 6
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2022-04-13 Classification: TRANSFERASE Ligands: CL, EKR |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-04-13
Ligands: CL, EKR
 |
Eed In Complex With Prc2 Allosteric Inhibitor Compound 7
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2022-04-13 Classification: TRANSFERASE Ligands: CL, EKF |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-04-13
Ligands: CL, EKF
 |
Eed In Complex With Prc2 Allosteric Inhibitor Compound 22 (Mak683)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2022-04-13 Classification: TRANSFERASE Ligands: CL, EJR |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-04-13
Ligands: CL, EJR
 |
Discovery Of Cdz173 (Leniolisib), Representing A Structurally Novel Class Of Pi3K Delta-Selective Inhibitors
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:2.90 Å Release Date: 2017-09-20 Classification: TRANSFERASE Ligands: 9NQ |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2017-09-20
Ligands: 9NQ
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Crystal Structure Of Pi3K Alpha With Pi3K Delta Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.02 Å Release Date: 2016-09-07 Classification: Transferase/Protein Transport/Inhibitor Ligands: 6CY |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-09-07
Ligands: 6CY
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Discovery Of Imidazoquinolines As A Novel Class Of Potent, Selective And In Vivo Efficacious Cot Kinase Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.70 Å Release Date: 2016-08-24 Classification: TRANSFERASE Ligands: 6DA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-08-24
Ligands: 6DA
 |
Discovery And Pharmacological Characterization Of Novel Quinazoline-Based Pi3K Delta-Selective Inhibitors
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:2.85 Å Release Date: 2016-08-10 Classification: TRANSFERASE Ligands: 6CY |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2016-08-10
Ligands: 6CY
 |
Co-Crystal Structure Of Lipid Kinase Pi3K Alpha With A Selective Phosphatidylinositol-3 Kinase Alpha Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.62 Å Release Date: 2016-05-18 Classification: transferase/transferase inhibitor Ligands: 4Q2 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-05-18
Ligands: 4Q2
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Syk Catalytic Domain Complexed With A Potent Orally Bioavailable Thiazole Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2015-09-23 Classification: Transferase/Transferase inhibitor Ligands: 55M |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-09-23
Ligands: 55M
 |
Syk Catalytic Domain Complexed With A Potent And Orally Bioavailable Benzisothiazole Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.76 Å Release Date: 2015-09-23 Classification: Transferase/Transferase inhibitor Ligands: 55Y |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-09-23
Ligands: 55Y
 |
Syk Catalytic Domain Complexed With Naphthyridine Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2015-09-16 Classification: Transferase/transferase inhibitor Ligands: GOL, CL, 55U |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-09-16
Ligands: GOL, CL, 55U
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Syk Catalytic Domain Complexed With A Potent Triazine Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2015-03-18 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: FMT, GOL, 3YV |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-03-18
Ligands: FMT, GOL, 3YV
 |
Syk Catalytic Domain Complexed With A Potent Triazine Inhibitor2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.59 Å Release Date: 2015-03-18 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: GOL, 3YX |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-03-18
Ligands: GOL, 3YX
 |
Syk Catalytic Domain Complexed With A Potent Pyrimidine Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.75 Å Release Date: 2015-03-18 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: GOL, 3YT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-03-18
Ligands: GOL, 3YT
 |
Syk Catalytic Domain In Complex With A Potent Pyridopyrimidinone Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2014-04-23 Classification: transferase/transferase inhibitor Ligands: 2X6 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-04-23
Ligands: 2X6
 |
Co-Crystal Structures Of The Lipid Kinase Pi3K Alpha With Pan And Isoform Selective Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2014-04-02 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: SCN, 1LT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-04-02
Ligands: SCN, 1LT