Search Count: 8
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Crystal Structure Of Jak1 Jh1 Domain In Complex With An Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.75 Å Release Date: 2024-11-06 Classification: SIGNALING PROTEIN Ligands: A1H5R, NA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-11-06
Ligands: A1H5R, NA
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Crystal Structure Of Rhodesain In Complex With A Macrolactam Inhibitor
Organism: Trypanosoma brucei rhodesiense
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2018-04-11 Classification: HYDROLASE Ligands: C2K, EDO |
Organism: Trypanosoma brucei rhodesiense
Method: X-RAY DIFFRACTION
Release Date: 2018-04-11
Ligands: C2K, EDO
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Crystal Structure Of Rhodesain In Complex With A Macrolactam Inhibitor
Organism: Trypanosoma brucei rhodesiense
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2018-04-11 Classification: HYDROLASE Ligands: EDO, C3E |
Organism: Trypanosoma brucei rhodesiense
Method: X-RAY DIFFRACTION
Release Date: 2018-04-11
Ligands: EDO, C3E
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Crystal Structure Of Rhodesain In Complex With A Macrolactam Inhibitor
Organism: Trypanosoma brucei rhodesiense
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2018-04-11 Classification: HYDROLASE Ligands: EDO, C2W |
Organism: Trypanosoma brucei rhodesiense
Method: X-RAY DIFFRACTION
Release Date: 2018-04-11
Ligands: EDO, C2W
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Cathepsin L In Complex With (3S,14E)-19-Chloro-N-(1-Cyanocyclopropyl)-5-Oxo-12,17-Dioxa-4-Azatricyclo[16.2.2.06,11]Docosa-1(21),6(11),7,9,14,18(22),19-Heptaene-3-Carboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.37 Å Release Date: 2018-04-11 Classification: HYDROLASE Ligands: C3E, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-04-11
Ligands: C3E, GOL
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Cathepsin L In Complex With (3S,14E)-19-Chloro-N-(1-Cyanocyclopropyl)-5-Oxo-17-Oxa-4-Azatricyclo[16.2.2.06,11]Docosa-1(21),6,8,10,14,18(22),19-Heptaene-3-Carboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.34 Å Release Date: 2018-04-11 Classification: HYDROLASE Ligands: C7Q |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-04-11
Ligands: C7Q
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Cathepsin L In Complex With (3S,14E)-8-(Azetidin-3-Yl)-19-Chloro-N-(1-Cyanocyclopropyl)-5-Oxo-12,17-Dioxa-4-Azatricyclo[16.2.2.06,11]Docosa-1(21),6,8,10,14,18(22),19-Heptaene-3-Carboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.02 Å Release Date: 2018-04-11 Classification: HYDROLASE Ligands: C7T, ZN, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-04-11
Ligands: C7T, ZN, CL
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Triazolopyridine Compounds As Selective Jak1 Inhibitors: From Hit Identification To Glpg0634
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2014-11-19 Classification: TRANSFERASE Ligands: 2HB |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-11-19
Ligands: 2HB
