Search Count: 11
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Usp7 In Complex With Gne6640 (4-(2-Amino-4-Ethyl-5-(1H-Indazol-5-Yl)Pyridin-3-Yl)Phenol)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.84 Å Release Date: 2017-10-25 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: 8JM |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-10-25
Ligands: 8JM
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Usp7 In Complex With Gne6776 (6'-Amino-4'-Ethyl-5'-(4-Hydroxyphenyl)-N-Methyl-[3,3'-Bipyridine]-6-Carboxamide)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.23 Å Release Date: 2017-10-25 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: 8JP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-10-25
Ligands: 8JP
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Crystal Structure Of P21-Activated Kinase 1 (Pak1) In Complex With Compound 9
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.22 Å Release Date: 2016-05-25 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 6BZ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-05-25
Ligands: 6BZ
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Cdk8/Cycc In Complex With Compound 20
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.39 Å Release Date: 2016-04-20 Classification: Transferase/Transcription Ligands: 66X, FMT, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-04-20
Ligands: 66X, FMT, CL
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Crystal Structure Of Cdk8:Cyclin C Complex With Compound 22
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.24 Å Release Date: 2016-02-10 Classification: Transcription/Transferase/Inhibitor Ligands: EDO, FMT, 50R |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-02-10
Ligands: EDO, FMT, 50R
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Crystal Structure Of Pak1 In Complex With An Inhibitor Compound G-5555
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2016-01-27 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 59T |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-01-27
Ligands: 59T
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Crystal Structure Of Pak1 In Complex With An Inhibitor Compound Frax1036
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2016-01-27 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 59U, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-01-27
Ligands: 59U, DMS
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Chk1 Kinase Domain With Diazacarbazole Compound 8: N-[3-(6-Cyano-9H-Pyrrolo[2,3-B:5,4-C']Dipyridin-3-Yl)Phenyl]Acetamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2015-06-03 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 3XK |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-06-03
Ligands: 3XK
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Chk1 Kinase Domain With Diazacarbazole Compound 7: 3-(2-Hydroxyphenyl)-9H-Pyrrolo[2,3-B:5,4-C']Dipyridine-6-Carbonitrile
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2015-06-03 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 3XL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-06-03
Ligands: 3XL
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Chk1 Kinase Domain With Diazacarbazole Compound 19
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.86 Å Release Date: 2015-06-03 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 3X7 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-06-03
Ligands: 3X7
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Crystal Structure Of Aurora-A In Complex With A Pentacyclic Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.70 Å Release Date: 2009-02-17 Classification: TRANSFERASE Ligands: 83H |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2009-02-17
Ligands: 83H
