Search Count: 13
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Rorcvar2 (Rorgt, 264-499) In Complex With Compound 1: Identification Of N-Aryl Imidazoles As Potent And Selective Rorgt Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.35 Å Release Date: 2019-11-27 Classification: TRANSCRIPTION Ligands: HJW |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-11-27
Ligands: HJW
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Rorcvar2 (Rorgt, 264-499) In Complex With Compound 2 At 2.3A: Identification Of N-Aryl Imidazoles As Potent And Selective Rorgt Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2019-11-27 Classification: TRANSCRIPTION Ligands: HKE, CHD |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-11-27
Ligands: HKE, CHD
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Rorcvar2 (Rorgt, 264-499) In Complex With Compound 4 At 2.2A: Identification Of N-Aryl Imidazoles As Potent And Selective Rorgt Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2019-11-27 Classification: TRANSCRIPTION Ligands: HKZ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-11-27
Ligands: HKZ
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Rorcvar2 (Rorgt, 264-499) In Complex With Compound 9 At 2.3A: Identification Of N-Aryl Imidazoles As Potent And Selective Rorgt Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2019-11-27 Classification: TRANSCRIPTION Ligands: HL8 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-11-27
Ligands: HL8
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Rorgt (264-518;C455S) In Complex With The Fragment ("Cpd-1") And Rip140 Peptide At 1.80A
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2018-07-18 Classification: TRANSCRIPTION Ligands: EE8 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-07-18
Ligands: EE8
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Rorgt (264-518;C455S) In Complex With Inverse Agonist "Cpd-2" And Rip140 Peptide At 1.90A
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2018-07-18 Classification: TRANSCRIPTION Ligands: EF5 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-07-18
Ligands: EF5
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Rorgt (264-518;C455S) In Complex With Inverse Agonist "Cpd-9" And Rip140 Peptide At 1.66A
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.66 Å Release Date: 2018-07-18 Classification: TRANSCRIPTION Ligands: EEZ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-07-18
Ligands: EEZ
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Lta4 Hydrolase (E297Q) Mutant In Complex With Pro-Gly-Pro Peptide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.84 Å Release Date: 2017-12-13 Classification: HYDROLASE Ligands: ZN, ACT, YB, IMD |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-12-13
Ligands: ZN, ACT, YB, IMD
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Lta4 Hydrolase In Complex With Compound11
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.95 Å Release Date: 2017-12-13 Classification: HYDROLASE Ligands: ZN, ACT, YB, IMD, BGW |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-12-13
Ligands: ZN, ACT, YB, IMD, BGW
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Lta4 Hydrolase In Complex With Compound15
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.24 Å Release Date: 2017-12-13 Classification: HYDROLASE Ligands: ZN, ACT, YB, IMD, BGK |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-12-13
Ligands: ZN, ACT, YB, IMD, BGK
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Synthesis And Biological Evaluation Of New Triazolo And Imidazolopyridine Rorgt Inverse Agonists
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.77 Å Release Date: 2016-12-14 Classification: TRANSCRIPTION Ligands: Q6Y |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-12-14
Ligands: Q6Y
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Crystal Structure Of Human Sphingosine-1-Phosphate Lyase In Complex With Inhibitor 6-[(2R)-4-(4-Benzyl-7-Chlorophthalazin-1-Yl)-2-Methylpiperazin-1-Yl]Pyridine-3-Carbonitrile
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2014-05-21 Classification: Lyase/Lyase inhibitor Ligands: SIN, GOL, 30J, PO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-05-21
Ligands: SIN, GOL, 30J, PO4
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Hiv-1 Protease In Complex With Sdz283-910
Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 1998-07-15 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: 2Z4 |
Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION
Release Date: 1998-07-15
Ligands: 2Z4