Search Count: 28
![]() |
Cryo-Em Structure Of The C. Neoformans Lipid Flippase Apt1-Cdc50 Bound With Butyrolactol A In The E2P State
Organism: Cryptococcus neoformans var. grubii h99
Method: ELECTRON MICROSCOPY Release Date: 2025-10-22 Classification: TRANSLOCASE/INHIBITOR Ligands: NAG, BEF, MG, A1BD6 |
Organism: Cryptococcus neoformans var. grubii h99
Method: ELECTRON MICROSCOPY
Release Date: 2025-10-22
Ligands: NAG, BEF, MG, A1BD6
![]() |
Crystal Structure Of Tnf Alpha In Complex With Compound 1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.36 Å Release Date: 2025-07-23 Classification: CYTOKINE Ligands: A1CB1 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-07-23
Ligands: A1CB1
![]() |
Crystal Structure Of Tnf Alpha In Complex With Compound 4
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2025-07-23 Classification: CYTOKINE Ligands: A1CB0 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-07-23
Ligands: A1CB0
![]() |
Crystal Structure Of Tnf Alpha In Complex With Compound 3.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.16 Å Release Date: 2025-07-23 Classification: CYTOKINE Ligands: A1CBZ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-07-23
Ligands: A1CBZ
![]() |
Crystal Structure Of Tnf Alpha In Complex With Compound 19
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.78 Å Release Date: 2025-07-23 Classification: CYTOKINE Ligands: A1CCE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-07-23
Ligands: A1CCE
![]() |
Crystal Structure Of The Human Pxr Ligand-Binding Domain In Complex With Furanodienone
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.95 Å Release Date: 2025-04-16 Classification: TRANSCRIPTION Ligands: XFQ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-04-16
Ligands: XFQ
![]() |
Cryo-Em Structure Of The C. Neoformans Lipid Flippase Apt1-Cdc50 In The E1 State
Organism: Cryptococcus neoformans var. grubii h99
Method: ELECTRON MICROSCOPY Release Date: 2025-02-05 Classification: LIPID TRANSPORT Ligands: NAG, MG |
Organism: Cryptococcus neoformans var. grubii h99
Method: ELECTRON MICROSCOPY
Release Date: 2025-02-05
Ligands: NAG, MG
![]() |
Crystal Structure Of Human Trf1 With Pinx1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.70 Å Release Date: 2024-09-04 Classification: DNA BINDING PROTEIN Ligands: HEZ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-09-04
Ligands: HEZ
![]() |
Il17A Homodimer Complexed To Compound 23
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.83 Å Release Date: 2024-04-03 Classification: CYTOKINE Ligands: XCE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-04-03
Ligands: XCE
![]() |
Il17A Complexed To Compound 7
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.47 Å Release Date: 2024-04-03 Classification: CYTOKINE Ligands: XCW, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-04-03
Ligands: XCW, CL
![]() |
Discovery Of Potent Myeloid Cell Leukemia-1 (Mcl-1) Inhibitors That Demonstrate In Vivo Activity In Mouse Xenograft Models Of Human Cancer
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2019-04-17 Classification: APOPTOSIS Ligands: KJP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-04-17
Ligands: KJP
![]() |
Novel Modes Of Inhibition Of Wild-Type Idh1: Direct Covalent Modification Of His315 With Cmpd1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.65 Å Release Date: 2018-07-25 Classification: OXIDOREDUCTASE/OXIDOREDUCTASE inhibitor Ligands: CA, ICT, DWP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-07-25
Ligands: CA, ICT, DWP
![]() |
Novel Binding Modes Of Inhibition Of Wild-Type Idh1: Allosteric Inhibition With Cmpd2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.17 Å Release Date: 2018-07-25 Classification: OXIDOREDUCTASE/OXIDOREDUCTASE inhibitor Ligands: LMR, MG, K32 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-07-25
Ligands: LMR, MG, K32
![]() |
Novel Modes Of Inhibition Of Wild-Type Idh1: Non-Equivalent Allosteric Inhibition With Cmpd3
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.01 Å Release Date: 2018-07-25 Classification: oxidoreductase/oxidoreductase inhibitor Ligands: NAP, DWM |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-07-25
Ligands: NAP, DWM
![]() |
Novel Modes Of Inhibition Of Wild-Type Idh1:Direct Covalent Modification Of His315 With Cmpd11
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.17 Å Release Date: 2018-07-25 Classification: OXIDOREDUCTASE/OXIDOREDUCTASE inhibitor Ligands: MG, ICT, DWJ, NAP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-07-25
Ligands: MG, ICT, DWJ, NAP
![]() |
Novel Modes Of Inhibition Of Wild-Type Idh1: Direct Covalent Modification Of His315 With Cmpd13
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.02 Å Release Date: 2018-07-25 Classification: oxidoreductase/oxidoreductase inhibitor Ligands: ICT, DWG, CA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-07-25
Ligands: ICT, DWG, CA
![]() |
Novel Modes Of Inhibition Of Wild-Type Idh1: Direct Covalent Modification Of His315 With Cmpd15
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.92 Å Release Date: 2018-07-25 Classification: oxidoreductase/oxidoreductase inhibitor Ligands: CA, ICT, DWS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-07-25
Ligands: CA, ICT, DWS
![]() |
Mcl-1 Complexed With Small Molecules
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.75 Å Release Date: 2018-01-31 Classification: APOPTOSIS Ligands: ECY |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-01-31
Ligands: ECY
![]() |
Mcl-1 Complexed With Small Molecules
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.90 Å Release Date: 2018-01-31 Classification: APOPTOSIS Ligands: ECM |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-01-31
Ligands: ECM
![]() |
Structure Of A Mcl-1 Inhibitor Binding To Site 3 Of Human Serum Albumin
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.70 Å Release Date: 2017-05-03 Classification: TRANSPORT PROTEIN Ligands: 6AK, PO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-05-03
Ligands: 6AK, PO4
