Search Count: 30
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Crystal Structure Of Human Ephrin Type-A Receptor 2 (Epha2) Kinase Domain In Complex With Jg165
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2023-11-22 Classification: TRANSFERASE Ligands: WT3, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-11-22
Ligands: WT3, EDO
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Human Mst3 (Stk24) Kinase In Complex With Macrocyclic Inhibitor Ja310
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.64 Å Release Date: 2023-11-08 Classification: TRANSFERASE Ligands: VY0, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-11-08
Ligands: VY0, EDO
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Human Mst3 (Stk24) Kinase In Complex With Inhibitor Mr24
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2023-11-08 Classification: TRANSFERASE Ligands: VYN, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-11-08
Ligands: VYN, EDO
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Human Mst3 (Stk24) Kinase In Complex With Inhibitor Mr26
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.61 Å Release Date: 2023-11-08 Classification: TRANSFERASE Ligands: VYH, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-11-08
Ligands: VYH, EDO
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Human Mst3 (Stk24) Kinase In Complex With Inhibitor Mr30
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.47 Å Release Date: 2023-11-08 Classification: TRANSFERASE Ligands: VZ2, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-11-08
Ligands: VZ2, EDO
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Crystal Structure Of The First Bromodomain Of Human Brd4 In Complex With The Dual Bet/Hdac Inhibitor Nb161
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.30 Å Release Date: 2023-07-05 Classification: GENE REGULATION Ligands: X9O, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-07-05
Ligands: X9O, EDO
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Crystal Structure Of The First Bromodomain Of Human Brd4 In Complex With The Dual Bet/Hdac Inhibitor Nb390
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.10 Å Release Date: 2023-07-05 Classification: GENE REGULATION Ligands: X9K, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-07-05
Ligands: X9K, EDO
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Crystal Structure Of The First Bromodomain Of Human Brd4 In Complex With The Dual Bet/Hdac Inhibitor Nb437
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.19 Å Release Date: 2023-07-05 Classification: GENE REGULATION Ligands: X9C, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-07-05
Ligands: X9C, EDO
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Crystal Structure Of The First Bromodomain Of Human Brd4 In Complex With The Dual Bet/Hdac Inhibitor Nb462
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.23 Å Release Date: 2023-07-05 Classification: GENE REGULATION Ligands: X8T, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-07-05
Ligands: X8T, EDO
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Crystal Structure Of The First Bromodomain Of Human Brd4 In Complex With The Dual Bet/Hdac Inhibitor Nb500
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.42 Å Release Date: 2023-07-05 Classification: GENE REGULATION Ligands: X8O, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-07-05
Ligands: X8O, EDO
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Crystal Structure Of The First Bromodomain Of Human Brd4 In Complex With The Dual Bet/Hdac Inhibitor Nb503
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.25 Å Release Date: 2023-07-05 Classification: GENE REGULATION Ligands: EDO, X9U |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-07-05
Ligands: EDO, X9U
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Crystal Structure Of The First Bromodomain Of Human Brd4 In Complex With The Dual Bet/Hdac Inhibitor Nb512
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.29 Å Release Date: 2023-07-05 Classification: GENE REGULATION Ligands: XA3, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-07-05
Ligands: XA3, EDO
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Human Mst3 (Stk24) Kinase In Complex With Inhibitor Mr39
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.72 Å Release Date: 2023-01-18 Classification: TRANSFERASE Ligands: SJL, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-01-18
Ligands: SJL, EDO
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Human Mst3 (Stk24) Kinase In Complex With Inhibitor Mrlw5
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.52 Å Release Date: 2023-01-18 Classification: TRANSFERASE Ligands: SJX, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-01-18
Ligands: SJX, EDO
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Crystal Structure Of Human Ephrin Type-A Receptor 2 (Epha2) Kinase Domain In Complex With Mr21
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.50 Å Release Date: 2022-11-23 Classification: TRANSFERASE Ligands: EDO, QRR |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-11-23
Ligands: EDO, QRR
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Crystal Structure Of Human Ephrin Type-A Receptor 2 (Epha2) Kinase Domain In Complex With Mral5
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2022-11-23 Classification: TRANSFERASE Ligands: EDO, QRD |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-11-23
Ligands: EDO, QRD
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The Stk17A (Drak1) Kinase Domain Bound To Ckjb68
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2022-02-02 Classification: TRANSFERASE Ligands: F7I |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-02-02
Ligands: F7I
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The Stk17A (Drak1) Kinase Domain Bound To Ck156
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2022-02-02 Classification: TRANSFERASE Ligands: F8I |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-02-02
Ligands: F8I
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Egfr(T790M/V948R) In Complex With Ln3844
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.76 Å Release Date: 2021-05-19 Classification: TRANSFERASE/TRANSFERASE inhibitor Ligands: UEJ, ANP, MG, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-05-19
Ligands: UEJ, ANP, MG, CL
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Crystal Structure Of Egfr(T790M/V948R) In Complex With Ln3753
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2021-03-31 Classification: TRANSFERASE Ligands: TOV, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-03-31
Ligands: TOV, CL
