Search Count: 188
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Discovery Of A Small Molecule Itk And Pan-Trk Kinase Inhibitor (Pf-07245303) For The Potential Topical Treatment Of Atopic Dermatitis
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.35 Å Release Date: 2025-11-19 Classification: SIGNALING PROTEIN Ligands: A1B66 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-11-19
Ligands: A1B66
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Cryo-Em Structure Of Ccr6 Bound By Pf-07054894 And Oxm2
Organism: Homo sapiens, Synthetic construct
Method: ELECTRON MICROSCOPY Resolution:3.35 Å Release Date: 2025-10-01 Classification: MEMBRANE PROTEIN Ligands: A1A1W, A1CH1 |
Organism: Homo sapiens, Synthetic construct
Method: ELECTRON MICROSCOPY
Release Date: 2025-10-01
Ligands: A1A1W, A1CH1
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Cryo-Em Structure Of Ttyh2 In Complex With Sybody 1 In Gdn
Organism: Homo sapiens, Vicugna pacos
Method: ELECTRON MICROSCOPY Release Date: 2025-05-21 Classification: MEMBRANE PROTEIN Ligands: NAG |
Organism: Homo sapiens, Vicugna pacos
Method: ELECTRON MICROSCOPY
Release Date: 2025-05-21
Ligands: NAG
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Cryo-Em Structure Of Ttyh2 In Complex With Lipids In Gdn
Organism: Homo sapiens
Method: ELECTRON MICROSCOPY Release Date: 2025-05-21 Classification: MEMBRANE PROTEIN Ligands: NAG, PLC, CLR, CPL |
Organism: Homo sapiens
Method: ELECTRON MICROSCOPY
Release Date: 2025-05-21
Ligands: NAG, PLC, CLR, CPL
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Cryo-Em Structure Of Ttyh3 In Gdn After Incubation With Apoe, Map2
Organism: Homo sapiens
Method: ELECTRON MICROSCOPY Release Date: 2025-05-21 Classification: MEMBRANE PROTEIN Ligands: NAG |
Organism: Homo sapiens
Method: ELECTRON MICROSCOPY
Release Date: 2025-05-21
Ligands: NAG
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Crystal Structure Of Melk With A Covalent Compound Gcl 99
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2025-03-05 Classification: TRANSFERASE Ligands: A1H9M |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-03-05
Ligands: A1H9M
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Crystal Structure Of Ulk1 With A Covalent Compound Gcl 99
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2025-01-08 Classification: TRANSFERASE Ligands: A1H9M |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-01-08
Ligands: A1H9M
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Crystal Structure Of Riok2 With A Covalent Compound Gcl 47
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.02 Å Release Date: 2025-01-08 Classification: TRANSFERASE Ligands: A1IBA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-01-08
Ligands: A1IBA
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Crystal Structure Of Ttbk1 With A Covalent Compound Gcl95
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.00 Å Release Date: 2025-01-08 Classification: TRANSFERASE Ligands: A1IU7 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-01-08
Ligands: A1IU7
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Cryo-Em Structure Of Ccr6 Bound By Sqa1 And Oxm2
Organism: Homo sapiens, Synthetic construct
Method: ELECTRON MICROSCOPY Release Date: 2024-09-11 Classification: MEMBRANE PROTEIN Ligands: CLR, EBX, A1A1W |
Organism: Homo sapiens, Synthetic construct
Method: ELECTRON MICROSCOPY
Release Date: 2024-09-11
Ligands: CLR, EBX, A1A1W
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Cryo-Em Structure Of Ccr6 Bound By Sqa1 And Oxm1
Organism: Homo sapiens, Synthetic construct
Method: ELECTRON MICROSCOPY Release Date: 2024-09-11 Classification: MEMBRANE PROTEIN Ligands: CLR, EBX, A1A2A |
Organism: Homo sapiens, Synthetic construct
Method: ELECTRON MICROSCOPY
Release Date: 2024-09-11
Ligands: CLR, EBX, A1A2A
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Structure Of Cul9-Rbx1 Ubiquitin E3 Ligase Complex - Hexameric Assembly
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Organism: Homo sapiens
Method: ELECTRON MICROSCOPY
Release Date: 2024-04-17
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Structure Of Cul9-Rbx1 Ubiquitin E3 Ligase Complex In Unneddylated And Neddylated Conformation - Focused Cullin Dimer
Organism: Homo sapiens
Method: ELECTRON MICROSCOPY Release Date: 2024-04-17 Classification: LIGASE Ligands: ZN |
Organism: Homo sapiens
Method: ELECTRON MICROSCOPY
Release Date: 2024-04-17
Ligands: ZN
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Structure Of Cul9-Rbx1 Ubiquitin E3 Ligase Complex In Unneddylated Conformation - Symmetry Expanded Unneddylated Dimer
Organism: Homo sapiens
Method: ELECTRON MICROSCOPY Release Date: 2024-04-17 Classification: LIGASE Ligands: ZN |
Organism: Homo sapiens
Method: ELECTRON MICROSCOPY
Release Date: 2024-04-17
Ligands: ZN
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Ubiquitin Ligation To Substrate By A Cullin-Ring E3 Ligase & Cdc34: Nedd8-Cul2-Rbx1-Elob/C-Fem1C With Trapped Ube2R2~Donor Ub-Sil1 Peptide
Organism: Homo sapiens
Method: ELECTRON MICROSCOPY Release Date: 2024-02-21 Classification: LIGASE Ligands: U9O, ZN |
Organism: Homo sapiens
Method: ELECTRON MICROSCOPY
Release Date: 2024-02-21
Ligands: U9O, ZN
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Ubiquitin Ligation To Neosubstrate By A Cullin-Ring E3 Ligase & Cdc34: Nedd8-Cul2-Rbx1-Elob/C-Vhl-Mz1 With Trapped Ube2R2~Donor Ub-Brd4 Bd2
Organism: Homo sapiens
Method: ELECTRON MICROSCOPY Release Date: 2024-02-21 Classification: LIGASE Ligands: ZN, SY8, 759 |
Organism: Homo sapiens
Method: ELECTRON MICROSCOPY
Release Date: 2024-02-21
Ligands: ZN, SY8, 759
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K48-Linked Ubiquitin Chain Formation With A Cullin-Ring E3 Ligase And Cdc34: Nedd8-Cul2-Rbx1-Elob/C-Fem1C With Trapped Ube2R2-Donor Ub-Acceptor Ub-Sil1 Peptide
Organism: Homo sapiens
Method: ELECTRON MICROSCOPY Release Date: 2024-02-14 Classification: LIGASE Ligands: SY8, ZN |
Organism: Homo sapiens
Method: ELECTRON MICROSCOPY
Release Date: 2024-02-14
Ligands: SY8, ZN
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Crystal Structure Of Human Ephrin Type-A Receptor 2 (Epha2) Kinase Domain In Complex With Jg165
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2023-11-22 Classification: TRANSFERASE Ligands: WT3, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-11-22
Ligands: WT3, EDO
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Human Mst3 (Stk24) Kinase In Complex With Macrocyclic Inhibitor Ja310
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.64 Å Release Date: 2023-11-08 Classification: TRANSFERASE Ligands: VY0, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-11-08
Ligands: VY0, EDO
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Human Mst3 (Stk24) Kinase In Complex With Inhibitor Mr24
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2023-11-08 Classification: TRANSFERASE Ligands: VYN, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-11-08
Ligands: VYN, EDO
