Search Count: 16
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Tubulin-7-Aminonoscapine Complex
Organism: Rattus norvegicus, Gallus gallus, Bos taurus
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2020-07-22 Classification: CELL CYCLE Ligands: GTP, MG, CA, GDP, OBQ, MES, GOL, ACP |
Organism: Rattus norvegicus, Gallus gallus, Bos taurus
Method: X-RAY DIFFRACTION
Release Date: 2020-07-22
Ligands: GTP, MG, CA, GDP, OBQ, MES, GOL, ACP
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Dual Inhibition Of The Essential Protein Kinases A And B In Mycobacterium Tuberculosis
Organism: Mycobacterium tuberculosis
Method: X-RAY DIFFRACTION Resolution:3.01 Å Release Date: 2018-02-14 Classification: TRANSFERASE/INHIBITOR Ligands: CJJ |
Organism: Mycobacterium tuberculosis
Method: X-RAY DIFFRACTION
Release Date: 2018-02-14
Ligands: CJJ
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Dual Inhibition Of The Essential Protein Kinases A And B In Mycobacterium Tuberculosis
Organism: Mycobacterium tuberculosis
Method: X-RAY DIFFRACTION Resolution:2.88 Å Release Date: 2018-02-14 Classification: TRANSFERASE/INHIBITOR Ligands: CJJ, 0BD |
Organism: Mycobacterium tuberculosis
Method: X-RAY DIFFRACTION
Release Date: 2018-02-14
Ligands: CJJ, 0BD
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Pb2 Bound To An Azaindole Inhibitor
Organism: Influenza a virus
Method: X-RAY DIFFRACTION Resolution:2.69 Å Release Date: 2017-05-17 Classification: RNA BINDING PROTEIN Ligands: 6NU |
Organism: Influenza a virus
Method: X-RAY DIFFRACTION
Release Date: 2017-05-17
Ligands: 6NU
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Pb2 Bound To An Azaindole Inhibitor
Organism: Influenza a virus
Method: X-RAY DIFFRACTION Resolution:2.93 Å Release Date: 2017-03-01 Classification: RNA BINDING PROTEIN Ligands: 6NS |
Organism: Influenza a virus
Method: X-RAY DIFFRACTION
Release Date: 2017-03-01
Ligands: 6NS
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Discovery Of Vx-509 (Decernotinib): A Potent And Selective Janus Kinase (Jak) 3 Inhibitor For The Treatment Of Autoimmune Disease
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.16 Å Release Date: 2015-08-12 Classification: Transferase/Transferase Inhibitor Ligands: 4HW |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-08-12
Ligands: 4HW
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Discovery Of Vx-509 (Decernotinib): A Potent And Selective Janus Kinase (Jak) 3 Inhibitor For The Treatment Of Autoimmune Diseases
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.78 Å Release Date: 2015-08-12 Classification: Transferase/Transferase Inhibitor Ligands: 4HZ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-08-12
Ligands: 4HZ
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Discovery Of Vx-509 (Decernotinib): A Potent And Selective Janus Kinase (Jak) 3 Inhibitor For The Treatment Of Autoimmune Diseases
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.04 Å Release Date: 2015-08-12 Classification: Transferase/Transferase Inhibitor Ligands: 467 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-08-12
Ligands: 467
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Discovery Of Vx-509 (Decernotinib): A Potent And Selective Janus Kinase (Jak) 3 Inhibitor For The Treatment Of Autoimmune Disease
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.52 Å Release Date: 2015-08-12 Classification: Transferase/Transferase Inhibitor Ligands: VJK |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-08-12
Ligands: VJK
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Influenza Polymerase Basic Protein 2 (Pb2) Bound To 7-Methyl-Gtp
Organism: Influenza a virus
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2014-07-30 Classification: TRANSCRIPTION/TRANSCRIPTION INHIBITOR Ligands: MGT, 11H |
Organism: Influenza a virus
Method: X-RAY DIFFRACTION
Release Date: 2014-07-30
Ligands: MGT, 11H
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Influenza Polymerase Basic Protein 2 (Pb2) Bound To A Small-Molecule Inhibitor
Organism: Influenza a virus
Method: X-RAY DIFFRACTION Resolution:2.82 Å Release Date: 2014-07-30 Classification: TRANSCRIPTION/TRANSCRIPTION INHIBITOR Ligands: 704 |
Organism: Influenza a virus
Method: X-RAY DIFFRACTION
Release Date: 2014-07-30
Ligands: 704
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Influenza A (Flu) Virus Polymerase Basic Protein 2 (Pb2) Bound To Vx787, An Azaindole Inhibitor
Organism: Influenza a virus
Method: X-RAY DIFFRACTION Resolution:2.52 Å Release Date: 2014-07-30 Classification: transferase/transferase inhibitor Ligands: 21G |
Organism: Influenza a virus
Method: X-RAY DIFFRACTION
Release Date: 2014-07-30
Ligands: 21G
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Janus Kinase 2 Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2009-12-01 Classification: TRANSFERASE Ligands: JZH, NA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2009-12-01
Ligands: JZH, NA
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A Novel Chemotype Of Kinase Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2009-11-24 Classification: TRANSFERASE Ligands: 3KC |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2009-11-24
Ligands: 3KC
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2-Aminopyrazolo[1,5-A]Pyrimidines As Potent And Selective Inhibitors Of Jak2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2009-11-10 Classification: TRANSFERASE Ligands: 1P5 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2009-11-10
Ligands: 1P5
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2-Aminopyrazolo[1,5-A]Pyrimidines As Potent And Selective Inhibitors Of Jak2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2009-11-10 Classification: TRANSFERASE Ligands: 1P6 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2009-11-10
Ligands: 1P6
