Search Count: 24
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Human M5 Muscarinic Acetylcholine Receptor Complex With Mini-Gq And Iperoxo
Organism: Homo sapiens, Rattus norvegicus
Method: ELECTRON MICROSCOPY Resolution:2.79 Å Release Date: 2025-10-08 Classification: MEMBRANE PROTEIN Ligands: IXO |
Organism: Homo sapiens, Rattus norvegicus
Method: ELECTRON MICROSCOPY
Release Date: 2025-10-08
Ligands: IXO
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Human M5 Muscarinic Acetylcholine Receptor Complex With Mini-Gq, Agonist Acetylcholine And Positive Allosteric Modulator Vu6007678
Organism: Lama glama, Rattus norvegicus, Homo sapiens, Mus musculus
Method: ELECTRON MICROSCOPY Resolution:2.06 Å Release Date: 2025-08-13 Classification: MEMBRANE PROTEIN Ligands: A1BKS, ACH |
Organism: Lama glama, Rattus norvegicus, Homo sapiens, Mus musculus
Method: ELECTRON MICROSCOPY
Release Date: 2025-08-13
Ligands: A1BKS, ACH
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Crystal Structure Of Stabilized A2A Adenosine Receptor A2Ar-Star2-Bril In Complex With Compound 7, A Novel Nanomolar A2A Receptor Antagonist From Modern Hit-Finding With Structure-Guided De Novo Design
Organism: Homo sapiens, Escherichia coli
Method: X-RAY DIFFRACTION Resolution:1.75 Å Release Date: 2025-06-18 Classification: MEMBRANE PROTEIN |
Organism: Homo sapiens, Escherichia coli
Method: X-RAY DIFFRACTION
Release Date: 2025-06-18
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Crystal Structure Of Stabilized A2A Adenosine Receptor A2Ar-Star2-Bril In Complex With Compound 9, A Novel Nanomolar A2A Receptor Antagonist From Modern Hit-Finding With Structure-Guided De Novo Design
Organism: Homo sapiens, Escherichia coli
Method: X-RAY DIFFRACTION Resolution:1.72 Å Release Date: 2025-06-18 Classification: MEMBRANE PROTEIN |
Organism: Homo sapiens, Escherichia coli
Method: X-RAY DIFFRACTION
Release Date: 2025-06-18
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Crystal Structure Of Sry Hmg Box Bound To Dna
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION Resolution:2.48 Å Release Date: 2024-09-25 Classification: DNA BINDING PROTEIN/DNA Ligands: EDO |
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION
Release Date: 2024-09-25
Ligands: EDO
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Solution Structure Of A Chimeric U2Af2 Rrm2 / Fubp1 N-Box
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Organism: Homo sapiens
Method: SOLUTION NMR
Release Date: 2023-07-26
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Btk1 Soaked With Compound 5, Y551 Is Sequestered
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.84 Å Release Date: 2021-05-19 Classification: TRANSFERASE Ligands: X9J, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-05-19
Ligands: X9J, DMS
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Btk1 Soaked With Compound 5, Y551 Is Sequestered
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.33 Å Release Date: 2021-05-19 Classification: TRANSFERASE Ligands: X9M |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-05-19
Ligands: X9M
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Btk1 Soaked With Compound 26
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.34 Å Release Date: 2021-05-19 Classification: TRANSFERASE Ligands: X9P, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-05-19
Ligands: X9P, DMS
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Btk1 Soaked With Compound 24
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.94 Å Release Date: 2021-05-19 Classification: TRANSFERASE Ligands: X9S, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-05-19
Ligands: X9S, DMS
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Btk1 Soaked With Compound 25
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.83 Å Release Date: 2021-05-19 Classification: TRANSFERASE Ligands: X9V, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-05-19
Ligands: X9V, DMS
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Btk1 Soaked With Compound 30
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.38 Å Release Date: 2021-05-19 Classification: TRANSFERASE Ligands: DMS, X9Y |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-05-19
Ligands: DMS, X9Y
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Discovery Of M5049: A Novel Selective Tlr7/8 Inhibitor For Treatment Of Autoimmunity
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.49 Å Release Date: 2020-12-30 Classification: IMMUNE SYSTEM Ligands: NAG, QLH, FMT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-12-30
Ligands: NAG, QLH, FMT
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Solution Structure Of U2Af2 Rrm1,2
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Organism: Homo sapiens
Method: SOLUTION NMR
Release Date: 2020-05-06
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Structure Of Human Bruton'S Tyrosine Kinase In Complex With Evobrutinib
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.41 Å Release Date: 2019-08-14 Classification: Transferase/Transferase Inhibitor Ligands: CL, MZJ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-08-14
Ligands: CL, MZJ
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Discovery Of Affinity-Based Probes For Btk Occupancy Assay
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.23 Å Release Date: 2019-02-06 Classification: IMMUNE SYSTEM Ligands: KHD |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-02-06
Ligands: KHD
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Btk In Complex With Gdc-0834
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.71 Å Release Date: 2017-05-24 Classification: TRANSFERASE Ligands: 2VL, EDO, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-05-24
Ligands: 2VL, EDO, GOL
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Structure Of Btk With Rn486
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.75 Å Release Date: 2017-05-24 Classification: TRANSFERASE Ligands: 7G6 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-05-24
Ligands: 7G6
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Btk1 Cocrystallized With Rn983
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.95 Å Release Date: 2017-05-24 Classification: TRANSFERASE Ligands: 7G7 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-05-24
Ligands: 7G7
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Btk1 Soaked With Ibrutinib-Rev
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.11 Å Release Date: 2017-05-24 Classification: TRANSFERASE Ligands: 1E8, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-05-24
Ligands: 1E8, DMS
