Search Count: 16
![]() |
Discovery Of Doravirine, An Orally Bioavailable Non-Nucleoside Reverse Transcriptase Inhibitor Potent Against A Wide Range Of Resistant Mutant Hiv Viruses
Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION Resolution:2.58 Å Release Date: 2014-02-12 Classification: Transferase/Inhhibitor, Hydrolase/Inhhibitor Ligands: 2KW |
Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION
Release Date: 2014-02-12
Ligands: 2KW
![]() |
Ptp1B In Complex With A Phosphonic Acid Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2008-06-10 Classification: HYDROLASE Ligands: MG, 825 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-06-10
Ligands: MG, 825
![]() |
A Mutant Rabbit Cathepsin K With A Nitrile Inhibitor
Organism: Oryctolagus cuniculus
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2006-03-07 Classification: HYDROLASE Ligands: NOQ |
Organism: Oryctolagus cuniculus
Method: X-RAY DIFFRACTION
Release Date: 2006-03-07
Ligands: NOQ
![]() |
Crystal Structure Of Caspase-3 With A Nicotinic Acid Aldehyde Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2004-05-11 Classification: HYDROLASE Ligands: NA3 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2004-05-11
Ligands: NA3
![]() |
Crystal Structure Of The Complex Of Caspase-3 With A Pryazinone Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2004-05-11 Classification: HYDROLASE Ligands: PZN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2004-05-11
Ligands: PZN
![]() |
Crystal Structure Of The Complex Of Caspase-3 With A Phenyl-Propyl-Ketone Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2004-05-11 Classification: HYDROLASE/HYDROLASE INHIBITOR |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2004-05-11
![]() |
Crystal Structure Of The Complex Of Caspase-3 With A Nicotinic Acid Aldehyde Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2004-05-11 Classification: HYDROLASE Ligands: NA4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2004-05-11
Ligands: NA4
![]() |
Crystal Structure Of The Complex Of Caspase-3 With A Bromomethoxyphenyl Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.00 Å Release Date: 2004-05-11 Classification: HYDROLASE/hydrolase inhibitor Ligands: 0ZZ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2004-05-11
Ligands: 0ZZ
![]() |
Crystal Structure Of The Complex Of Caspase-3 With A Cinnamic Acid Methyl Ester Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.00 Å Release Date: 2004-05-11 Classification: HYDROLASE Ligands: CNE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2004-05-11
Ligands: CNE
![]() |
Crystal Structure Of The Complex Of Caspase-3 With A 5,6,7 Tricyclic Peptidomimetic Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.51 Å Release Date: 2004-05-11 Classification: HYDROLASE Ligands: 3CY |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2004-05-11
Ligands: 3CY
![]() |
The Structure Of Phosphotyrosine Phosphatase 1B In Complex With Compound 2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2003-09-30 Classification: HYDROLASE Ligands: 335 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2003-09-30
Ligands: 335
![]() |
The Structure Of Phosphotyrosine Phosphatase 1B In Complex With Compound 3
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2003-09-30 Classification: HYDROLASE Ligands: P27 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2003-09-30
Ligands: P27
![]() |
The Structure Of Phosphotyrosine Phosphatase 1B In Complex With Compound 4
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2003-09-30 Classification: HYDROLASE Ligands: MG, CL, P90 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2003-09-30
Ligands: MG, CL, P90
![]() |
The Structure Of Phosphotyrosine Phosphatase 1B In Complex With Compound 6
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2003-09-30 Classification: HYDROLASE Ligands: CL, 213 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2003-09-30
Ligands: CL, 213
![]() |
The Structure Of Phosphotyrosine Phosphatase 1B In Complex With Compound 9
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2003-09-30 Classification: HYDROLASE Ligands: CL, MG, 214, MPD |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2003-09-30
Ligands: CL, MG, 214, MPD
![]() |
The Structure Of Phosphotyrosine Phosphatase 1B In Complex With Compound 11
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2003-09-30 Classification: HYDROLASE Ligands: MG, 600 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2003-09-30
Ligands: MG, 600
