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Search Count: 10

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7LUK image
Crystal Structure Of Rar-Related Orphan Receptor C (Nhis-Rorgt(244-487)-L6-Src1(678-692) In Complex With An Azatricyclic Rorgt Inverse Agonist
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.09 Å Release Date: 2021-05-12
Classification: TRANSFERASE
Ligands: YDY

7JYM image
Crystal Structure Of Rar-Related Orphan Receptor C (Nhis-Rorgt(244-487)-L6-Src1(678-692)) In Complex With A Tricyclic Sulfone Inverse Agonist

6VQF image
Crystal Structure Of Rar-Related Orphan Receptor C (Nhis-Rorgt(244- 487)-L6-Src1(678-692)) In Complex With An Inverse Agonist

6U25 image
Crystal Structure Of Rar-Related Orphan Receptor C (Nhis- Rorgt(244-487)-L6-Src1(678-692)) In Complex With A Tricyclic Inverse Agonist

6O8I image
Btk In Complex With Inhibitor

5VLR image
Crystal Structure Of Pi3K Delta In Complex With A Trifluoro-Ethyl-Pyrazol-Pyrolotriazine Inhibitor

5T18 image
Crystal Structure Of Bruton Agammabulinemia Tyrosine Kinase Complexed With Bms-986142 Aka (2S)-6-Fluoro-5-[3-(8-Fluoro-1-Methyl-2,4-Dioxo-1,2,3,4-Tetrahydroquinazolin-3-Yl)-2-Methylphenyl]-2-(2-Hydroxypropan-2-Yl)-2,3,4,9-Tetrahydro-1H-Carbazole-8-Carboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.50 Å Release Date: 2017-03-08
Classification: TRANSFERASE
Ligands: 73T

5JRS image
Crystal Structure Of Bruton Agammaglobulinemia Tyrosine Kinase Complexed With 4-[2-Fluoro-3-(4-Oxo -3,4-Dihydroquinazolin-3-Yl)Phenyl]-7-(2-Hydroxypropan-2-Y L)-9H-Carbazole-1-Carboxamide

5BPY image
Crystal Structure Of Bruton Agammaglobulinemia Tyrosine Kinase Complexed With Bms-824171 Aka 6-[(3R)-3-(4-Tert-Bu Tylbenzamido)Piperidin-1-Yl]-2-{[4-(Morpholine-4-Carbonyl) Phenyl]Amino}Pyridine-3-Carboxamide

5BQ0 image
Crystal Structure Of Bruton Agammaglobulinemia Tyrosine Kinase Complexed With Bms-824171 Aka 6-[(3R)-3-(4-Tert-Bu Tylbenzamido)Piperidin-1-Yl]-2-{[4-(Morpholine-4-Carbonyl) Phenyl]Amino}Pyridine-3-Carboxamide
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