Search Count: 18
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Cryo-Em Structure Of Alk In Complex With Crbn/Ddb1 And Tri-611
Organism: Homo sapiens
Method: ELECTRON MICROSCOPY Release Date: 2026-08-05 Classification: LIGASE Ligands: ZN, A1CRM |
Organism: Homo sapiens
Method: ELECTRON MICROSCOPY
Release Date: 2026-08-05
Ligands: ZN, A1CRM
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Human Steroidogenic Cytochrome P450 17A1 With 3-Keto-5Alpha-Abiraterone Analog
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.01 Å Release Date: 2021-05-26 Classification: OXIDOREDUCTASE Ligands: HEM, UDJ, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-05-26
Ligands: HEM, UDJ, CL
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Human Steroidogenic Cytochrome P450 17A1 With 3-Keto-Delta4-Abiraterone Analog
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.70 Å Release Date: 2021-05-05 Classification: OXIDOREDUCTASE Ligands: HEM, U7P, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-05-05
Ligands: HEM, U7P, CL
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Human Steroidogenic Cytochrome P450 17A1 Mutant N52Y With Inhibitor Abiraterone
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2021-05-05 Classification: OXIDOREDUCTASE Ligands: HEM, AER |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-05-05
Ligands: HEM, AER
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Structure Of Human Cytochrome P450 1A1 With Duocarmycin Prodrug (S) Ict-2700
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.85 Å Release Date: 2020-09-23 Classification: OXIDOREDUCTASE Ligands: HEM, Q4M |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-09-23
Ligands: HEM, Q4M
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Structure Of Human Cytochrome P450 1A1 With Duocarmycin Prodrug (S) Ict-2726
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.08 Å Release Date: 2020-09-23 Classification: OXIDOREDUCTASE Ligands: HEM, Q4P, CPS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-09-23
Ligands: HEM, Q4P, CPS
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Structure Of An Ancestral-Reconstructed Cytochrome P450 1B1 With Alpha-Naphthoflavone
Organism: Synthetic construct
Method: X-RAY DIFFRACTION Resolution:2.95 Å Release Date: 2020-03-18 Classification: OXIDOREDUCTASE Ligands: BHF, HEM, GOL |
Organism: Synthetic construct
Method: X-RAY DIFFRACTION
Release Date: 2020-03-18
Ligands: BHF, HEM, GOL
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Structure Of An Ancestral-Reconstructed Cytochrome P450 1B1 With Estradiol
Organism: Synthetic construct
Method: X-RAY DIFFRACTION Resolution:3.10 Å Release Date: 2020-03-18 Classification: OXIDOREDUCTASE Ligands: EST, HEM |
Organism: Synthetic construct
Method: X-RAY DIFFRACTION
Release Date: 2020-03-18
Ligands: EST, HEM
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Structure Of Human Cytochrome P450 1A1 With 5-Amino-N-(5-((4R,5R)-4-Amino-5-Fluoroazepan-1-Yl)-1-Methyl-1H-Pyrazol-4-Yl)-2-(2,6-Difluorophenyl)Thiazole-4-Carboxamide)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.17 Å Release Date: 2019-12-04 Classification: OXIDOREDUCTASE Ligands: HEM, KUV, NO3 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-12-04
Ligands: HEM, KUV, NO3
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Structure Of Human Cytochrome P450 1A1 With Bergamottin
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.85 Å Release Date: 2018-10-03 Classification: OXIDOREDUCTASE Ligands: HEM, HJJ, CPS, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-10-03
Ligands: HEM, HJJ, CPS, GOL
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Structure Of Human Cytochrome P450 1A1 With Erlotinib
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.00 Å Release Date: 2018-10-03 Classification: OXIDOREDUCTASE Ligands: HEM, AQ4, CPS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-10-03
Ligands: HEM, AQ4, CPS
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Human Steroidogenic Cytochrome P450 17A1 With 3Alphaoh-5Alpha-Abiraterone Analog
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.39 Å Release Date: 2018-02-28 Classification: OXIDOREDUCTASE Ligands: HEM, 8QD |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-02-28
Ligands: HEM, 8QD
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Crystal Structure Of Hpnmt In Complex With Bisubstrate Inhibitor N-(3-((((2S,3S,4R,5R)-5-(6-Amino-9H-Purin-9-Yl)-3,4-Dihydroxytetrahydrofuran-2-Yl)Methyl)Thio)Propyl)-1,2,3,4-Tetrahydroisoquinoline-3-Carboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2014-10-15 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 2D5, TRS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-10-15
Ligands: 2D5, TRS
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Crystal Structure Of Hpnmt In Complex With Bisubstrate Inhibitor (2R,3R,4S,5S)-2-(6-Amino-9H-Purin-9-Yl)-5-(((2-(((7-Nitro-1,2,3,4-Tetrahydroisoquinolin-3-Yl)Methyl)Amino)Ethyl)Thio)Methyl)Tetrahydrofuran-3,4-Diol
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.95 Å Release Date: 2014-09-10 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: JIL, TRS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-09-10
Ligands: JIL, TRS
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Human Cytochrome P450 2A6 I208S/I300F/G301A/S369G In Complex With Pilocarpine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2011-12-07 Classification: OXIDOREDUCTASE Ligands: HEM, 9PL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-12-07
Ligands: HEM, 9PL
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Human Cytochrome P450 2A6 In Complex With Pilocarpine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2011-12-07 Classification: OXIDOREDUCTASE Ligands: HEM, 9PL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-12-07
Ligands: HEM, 9PL
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Human Cytochrome P450 2A13 In Complex With Pilocarpine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.00 Å Release Date: 2011-12-07 Classification: OXIDOREDUCTASE Ligands: HEM, 9PL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-12-07
Ligands: HEM, 9PL
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Human Cytochrome P450 2E1 In Complex With Pilocarpine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.35 Å Release Date: 2011-12-07 Classification: OXIDOREDUCTASE Ligands: HEM, 9PL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-12-07
Ligands: HEM, 9PL
