Search Count: 13
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Crystal Structure Of Egfr Double Mutant (T790M/L858R) In Complex With Compound 6.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.56 Å Release Date: 2021-10-20 Classification: TRANSFERASE Ligands: 35Z |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-10-20
Ligands: 35Z
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Novel Atp-Competitive Mk2 Inhibitors With Potent Biochemical And Cell-Based Activity Throughout The Series
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.25 Å Release Date: 2011-12-14 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: I85 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-12-14
Ligands: I85
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Mk3 Kinase Bound To Compound 5B
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.09 Å Release Date: 2011-05-25 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 05B |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-05-25
Ligands: 05B
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Mk2 Kinase Bound To Compound 5B
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.90 Å Release Date: 2011-05-25 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 05B |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-05-25
Ligands: 05B
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Mk2 Kinase Bound To Compound 1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.00 Å Release Date: 2011-05-25 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: MLI, P4O |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-05-25
Ligands: MLI, P4O
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Mk2 Kinase Bound To Compound 2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.20 Å Release Date: 2011-05-25 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: CD2 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-05-25
Ligands: CD2
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Drug Resistant Csrc Kinase Domain In Complex With Covalent Inhibitor Pd168393
Organism: Gallus gallus
Method: X-RAY DIFFRACTION Resolution:2.48 Å Release Date: 2010-12-22 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: DJK |
Organism: Gallus gallus
Method: X-RAY DIFFRACTION
Release Date: 2010-12-22
Ligands: DJK
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N-Benzyl-Indolo Carboxylic Acids: Design And Synthesis Of Potent And Selective Adipocyte Fatty-Acid Binding Protein (A-Fabp) Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2009-03-10 Classification: LIPID BINDING PROTEIN Ligands: 8CA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2009-03-10
Ligands: 8CA
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N-Benzyl-Indolo Carboxylic Acids: Design And Synthesis Of Potent And Selective Adipocyte Fatty-Acid Binding Protein (A-Fabp) Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.16 Å Release Date: 2009-03-10 Classification: LIPID BINDING PROTEIN Ligands: F8A |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2009-03-10
Ligands: F8A
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N-Benzyl-Indolo Carboxylic Acids: Design And Synthesis Of Potent And Selective Adipocyte Fatty-Acid Binding Protein (A-Fabp) Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2009-03-10 Classification: LIPID BINDING PROTEIN Ligands: I4A |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2009-03-10
Ligands: I4A
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Crystal Structure Of Human Adipocyte Fatty Acid Binding Protein In Complex With A Non-Covalent Ligand
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2004-08-24 Classification: LIPID TRANSPORT Ligands: B1V |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2004-08-24
Ligands: B1V
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Crystal Structure Of Human Adipocyte Fatty Acid Binding Protein In Complex With A Carboxylic Acid Ligand
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2004-08-24 Classification: LIPID TRANSPORT Ligands: CRZ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2004-08-24
Ligands: CRZ
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Human Ptp1B Catalytic Domain Complexed With Pnu177836
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2002-02-13 Classification: HYDROLASE Ligands: TBH |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2002-02-13
Ligands: TBH
