Search Count: 46
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Human Cdk8/Cyclin-C Complex With Inhibitor 2-9
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.57 Å Release Date: 2025-01-22 Classification: TRANSCRIPTION Ligands: EDO, GOL, A1IS8, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-01-22
Ligands: EDO, GOL, A1IS8, DMS
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Human Cdk8/Cyclin-C Complex With Inhibitor 3-7
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.16 Å Release Date: 2025-01-22 Classification: TRANSCRIPTION Ligands: CL, EDO, GOL, A1ITF, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-01-22
Ligands: CL, EDO, GOL, A1ITF, DMS
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Mycobacterium Tuberculosis 3-Hydroxyl-Acp Dehydratase Hadab In Complex With 1,3-Diarylpyrazolyl-Acylsulfonamide Inhibitor
Organism: Mycobacterium tuberculosis
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2022-11-16 Classification: LYASE/INHIBITOR Ligands: CI7, EDO, PEG, GOL |
Organism: Mycobacterium tuberculosis
Method: X-RAY DIFFRACTION
Release Date: 2022-11-16
Ligands: CI7, EDO, PEG, GOL
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N-Terminal Bromodomain Of Human Brd4 With Compound 3Ag
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.17 Å Release Date: 2021-10-06 Classification: TRANSCRIPTION Ligands: 5Z4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-10-06
Ligands: 5Z4
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N-Terminal Bromodomain Of Human Brd4 With Compound 3Bg
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.31 Å Release Date: 2021-10-06 Classification: TRANSCRIPTION Ligands: 5YY |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-10-06
Ligands: 5YY
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N-Terminal Bromodomain Of Human Brd4 With Compound 5Ef
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.88 Å Release Date: 2021-10-06 Classification: TRANSCRIPTION Ligands: 5Z1 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-10-06
Ligands: 5Z1
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Fak Protac Gsk215 In Complex With Fak And Pvhl:Elonginc:Elonginb
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.24 Å Release Date: 2021-09-29 Classification: TRANSFERASE Ligands: 7QB, PEG, EDO, CA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-09-29
Ligands: 7QB, PEG, EDO, CA
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Human Dnmt1(729-1600) Bound To Zebularine-Containing 12Mer Dsdna
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2021-07-07 Classification: TRANSFERASE Ligands: SAH, ZN, EDO, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-07-07
Ligands: SAH, ZN, EDO, GOL
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Human Dnmt1(729-1600) Bound To Zebularine-Containing 12Mer Dsdna And Inhibitor Gsk3830052
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.79 Å Release Date: 2021-07-07 Classification: TRANSFERASE/TRANSFERASE INHIBITOR/DNA Ligands: ZN, EDO, X52 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-07-07
Ligands: ZN, EDO, X52
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Human Dnmt1(729-1600) Bound To Zebularine-Containing 12Mer Dsdna And Inhibitor Gsk3685032A
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.65 Å Release Date: 2021-07-07 Classification: TRANSFERASE/TRANSFERASE INHIBITOR/DNA Ligands: ZN, EDO, UXM |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-07-07
Ligands: ZN, EDO, UXM
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N-Terminal Bromodomain Of Human Brd4 With Ibet-Bd1 (Gsk778)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.28 Å Release Date: 2020-04-01 Classification: TRANSCRIPTION Ligands: GLU, LWB, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-04-01
Ligands: GLU, LWB, EDO
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C-Terminal Bromodomain Of Human Brd2 With Ibet-Bd1 (Gsk778)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2020-04-01 Classification: TRANSCRIPTION Ligands: LWB, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-04-01
Ligands: LWB, EDO
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C-Terminal Bromodomain Of Human Brd2 With Ibet-Bd2 (Gsk046)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2020-04-01 Classification: TRANSCRIPTION Ligands: EDO, LW5 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-04-01
Ligands: EDO, LW5
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N-Terminal Bromodomain Of Human Brd4 With Ibet-Bd2 (Gsk046)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2020-04-01 Classification: TRANSCRIPTION Ligands: EDO, LW5 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-04-01
Ligands: EDO, LW5
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Pi3K Delta In Complex With N[5(7{2[4(2Hydroxypropan2Yl)Piperidin1 Yl]Ethoxy}1,3Dihydro2Benzofuran5Yl)2 Methoxypyridin3Yl]Methanesulfonamide
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2020-01-01 Classification: TRANSFERASE Ligands: NQ2 |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2020-01-01
Ligands: NQ2
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Pi3K Delta In Complex With 2Methoxyn[2Methoxy5(7{[(2R)4(Oxetan3 Yl)Morpholin2Yl]Methoxy}1,3Dihydro2 Benzofuran5Yl)Pyridin3Yl]Ethane1 Sulfonamide
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2020-01-01 Classification: TRANSFERASE Ligands: NQ5 |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2020-01-01
Ligands: NQ5
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Amidobenzimidazole (Abzi) Sting Agonists
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.91 Å Release Date: 2018-11-07 Classification: immune system/agonist Ligands: CA, HGJ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-11-07
Ligands: CA, HGJ
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Linked Amidobenzimidazole Sting Agonist
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.45 Å Release Date: 2018-11-07 Classification: immune system/agonist Ligands: HG4, CA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-11-07
Ligands: HG4, CA
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Pi3 Kinase Delta In Complex With Methyl 5-(4-(5-((4-Isopropylpiperazin-1-Yl)Methyl)Oxazol-2-Yl)-1H-Indazol-6-Yl)-2-Methoxynicotinate
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:2.04 Å Release Date: 2017-12-27 Classification: TRANSFERASE Ligands: C5Z |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2017-12-27
Ligands: C5Z
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Pi3 Kinase Delta In Complex With 4-Fluorophenyl 5-(4-(5-((4-Isopropylpiperazin-1-Yl)Methyl)Oxazol-2-Yl)-1H-Indazol-6-Yl)-2-Methoxynicotinate
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2017-12-20 Classification: TRANSFERASE Ligands: C5W |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2017-12-20
Ligands: C5W
