Search Count: 10
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Crystal Structure Of Alpha-V Beta-1 Integrin Headpiece In Complex With Tr01225179
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.45 Å Release Date: 2025-01-01 Classification: CELL ADHESION Ligands: CA, NAG, A1AFA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-01-01
Ligands: CA, NAG, A1AFA
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Fragment-Based Discovery Of A Novel Bruton'S Tyrosine Kinase Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.25 Å Release Date: 2021-09-08 Classification: TRANSFERASE/TRANSFERASE inhibitor Ligands: IMD, PGO, 0BQ, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-09-08
Ligands: IMD, PGO, 0BQ, EDO
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Fragment-Based Discovery Of A Novel Bruton'S Tyrosine Kinase Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.55 Å Release Date: 2021-09-08 Classification: TRANSFERASE/TRANSFERASE inhibitor Ligands: IMD, EDO, DMS, 0UW |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-09-08
Ligands: IMD, EDO, DMS, 0UW
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Fragment-Based Discovery Of A Novel Bruton'S Tyrosine Kinase Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2021-09-08 Classification: TRANSFERASE/TRANSFERASE inhibitor Ligands: IMD, PGO, DMS, 0GW |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-09-08
Ligands: IMD, PGO, DMS, 0GW
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Fragment-Based Drug Design Of A Novel, Covalent Bruton'S Tyrosine Kinase Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2021-09-08 Classification: TRANSFERASE/TRANSFERASE inhibitor Ligands: IMD, 0CI, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-09-08
Ligands: IMD, 0CI, DMS
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Met Tyrosine Kinase Inhibition Enhances The Antitumor Efficacy Of An Hgf Antibody
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2020-02-12 Classification: TRANSFERASE-TRANSFERASE INHIBITOR Ligands: 84S, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-02-12
Ligands: 84S, CL
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Met Tyrosine Kinase Inhibition Enhances The Antitumor Efficacy Of An Hgf Antibody
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2017-05-31 Classification: TRANSFERASE/INHIBITOR Ligands: 84M, GOL, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-05-31
Ligands: 84M, GOL, CL
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Met Tyrosine Kinase Inhibition Enhances The Antitumor Efficacy Of An Hgf Antibody
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.25 Å Release Date: 2017-05-31 Classification: TRANSFERASE/INHIBITOR Ligands: 84P, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-05-31
Ligands: 84P, CL
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Structure-Based Optimization Of 1H-Imidazole-2-Carboxamides As Axl Kinase Inhibitors Utilizing A Mer Mutant Surrogate
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.24 Å Release Date: 2017-01-25 Classification: Transferase/Transferase Inhibitor Ligands: 79Y |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-01-25
Ligands: 79Y
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Structure-Based Optimization Of 1H-Imidazole-2-Carboxamides As Axl Kinase Inhibitors Utilizing A Mer Mutant Surrogate
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.68 Å Release Date: 2017-01-25 Classification: Transferase/Transferase Inhibitor Ligands: 7AE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-01-25
Ligands: 7AE
