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6ODA image
Crystal Structure Of Hdac8 In Complex With Compound 2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.88 Å Release Date: 2020-04-01
Classification: HYDROLASE
Ligands: C7, ZN, K

6ODB image
Crystal Structure Of Hdac8 In Complex With Compound 3
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.70 Å Release Date: 2020-04-01
Classification: HYDROLASE
Ligands: M8G, ZN, K, GOL

6ODC image
Crystal Structure Of Hdac8 In Complex With Compound 30
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.80 Å Release Date: 2020-04-01
Classification: HYDROLASE
Ligands: ZN, K, M7Y, EDO

6P3P image
Crystal Structure Of Mcl-1 In Complex With Compound 65

6O2Y image
Crystal Structure Of Idh1 R132H Mutant In Complex With Compound 24

6O2Z image
Crystal Structure Of Idh1 R132H Mutant In Complex With Compound 32

6NNA image
Human Fatty Acid Synthase Psi/Kr Tri-Domain With Nadph And Compound 22
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.26 Å Release Date: 2019-02-20
Classification: TRANSFERASE
Ligands: NDP, KUA, EDO

5NGE image
Crystal Structure Of Usp7 In Complex With The Non-Covalent Inhibitor, Ft671
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.35 Å Release Date: 2017-10-18
Classification: HYDROLASE
Ligands: 8WK

5NGF image
Crystal Structure Of Usp7 In Complex With The Covalent Inhibitor, Ft827
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.33 Å Release Date: 2017-10-18
Classification: HYDROLASE
Ligands: 8WN, EDO

5KIT image
Crystal Structure Of Nicotinamide Phosphoribosyltransferase (Nampt) In Complex With Inhibitors 37

4WQ6 image
The Crystal Structure Of Human Nicotinamide Phosphoribosyltransferase (Nampt) In Complex With N-(4-{(S)-[1-(2-Methylpropyl)Piperidin-4-Yl]Sulfinyl}Benzyl)Furo[2,3-C]Pyridine-2-Carboxamide Inhibitor (Compound 21)

4O13 image
The Crystal Structure Of Nampt In Complex With Gne-618

4O14 image
Structural Basis For Resistance To Diverse Classes Of Nampt Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.87 Å Release Date: 2014-10-22
Classification: TRANSFERASE
Ligands: PO4, EDO

4O15 image
The Crystal Structure Of A Mutant Nampt (S165F) In Complex With Gne-618

4O16 image
Structural Basis For Resistance To Diverse Classes Of Nampt Inhibitors

4O17 image
Structural Basis For Resistance To Diverse Classes Of Nampt Inhibitors

4O18 image
Structural Basis For Resistance To Diverse Classes Of Nampt Inhibitors

4O19 image
The Crystal Structure Of A Mutant Nampt (G217V)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.75 Å Release Date: 2014-10-22
Classification: TRANSFERASE
Ligands: PO4, EDO

4O1A image
The Crystal Structure Of The Mutant Nampt G217R

4O1B image
The Crystal Structure Of A Mutant Nampt (G217R) In Complex With An Inhibitor Apo866
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