Search Count: 10
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Crystal Structure Of Braf Kinase Domain With Pf-07284890
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.92 Å Release Date: 2024-08-14 Classification: SIGNALING PROTEIN Ligands: PEG, GOL, A1AN9 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-08-14
Ligands: PEG, GOL, A1AN9
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Identification Of The Clinical Development Candidate Mrtx849, A Covalent Krasg12C Inhibitor For The Treatment Of Cancer
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.27 Å Release Date: 2020-04-22 Classification: HYDROLASE/INHIBITOR Ligands: GDP, MG, M1R |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-04-22
Ligands: GDP, MG, M1R
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Identification Of The Clinical Development Candidate Mrtx849, A Covalent Krasg12C Inhibitor For The Treatment Of Cancer
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.03 Å Release Date: 2020-04-22 Classification: HYDROLASE/INHIBITOR Ligands: GDP, MG, QH4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-04-22
Ligands: GDP, MG, QH4
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Identification Of The Clinical Development Candidate Mrtx849, A Covalent Krasg12C Inhibitor For The Treatment Of Cancer
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.94 Å Release Date: 2020-04-22 Classification: HYDROLASE/INHIBITOR Ligands: GDP, MG, M1X |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-04-22
Ligands: GDP, MG, M1X
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Crystal Structure Of Glucokinase In Complex With Compound 6
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.70 Å Release Date: 2019-07-10 Classification: Transferase/Transferase Inhibitor Ligands: GLC, HKM |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-07-10
Ligands: GLC, HKM
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Crystal Structure Of Glucokinase In Complex With Compound 72
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2019-07-10 Classification: Transferase/Transferase Inhibitor Ligands: GLC, DMS, HKG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-07-10
Ligands: GLC, DMS, HKG
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Tetrahydropyridopyrimidines As Covalent Inhibitors Of Kras-G12C
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2018-12-12 Classification: ONCOPROTEIN Ligands: GDP, MG, K9M |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-12-12
Ligands: GDP, MG, K9M
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Tetrahydropyridopyrimidines As Covalent Inhibitors Of Kras-G12C
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.72 Å Release Date: 2018-12-12 Classification: ONCOPROTEIN Ligands: GDP, MG, K9J |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-12-12
Ligands: GDP, MG, K9J
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Structure Of Cytochrome P450 4B1 (Cyp4B1) Complexed With Octane: An N-Alkane And Fatty Acid Omega-Hydroxylase With A Covalently Bound Heme
Organism: Oryctolagus cuniculus
Method: X-RAY DIFFRACTION Resolution:2.70 Å Release Date: 2017-02-15 Classification: OXIDOREDUCTASE Ligands: HEM, OCT |
Organism: Oryctolagus cuniculus
Method: X-RAY DIFFRACTION
Release Date: 2017-02-15
Ligands: HEM, OCT
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Discovery Of 2-Pyridyl Ureas As Glucokinase Activators
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2014-10-08 Classification: TRANSFERASE Ligands: GLC, 3LZ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-10-08
Ligands: GLC, 3LZ
