Search Count: 5
![]() |
Crystal Structure Of Rorgt With 3-Cyano-N-(3-{[(3S)-4-(Cyclopentanecarbonyl)-3-Methylpiperazin-1-Yl]Methyl}-5-Fluoro-2-Methylphenyl)Benzamide (Compound 1)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2020-03-04 Classification: PROTEIN BINDING Ligands: LKY, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-03-04
Ligands: LKY, EDO
![]() |
Structure Of Focal Adhesion Kinase Catalytic Domain In Complex With Hinge Binding Pyrazolobenzothiazine Compound.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.55 Å Release Date: 2013-03-06 Classification: transferase/transferase inhibitor Ligands: 1BQ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-03-06
Ligands: 1BQ
![]() |
Structure Of Focal Adhesion Kinase Catalytic Domain In Complex With An Allosteric Binding Pyrazolobenzothiazine Compound.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.75 Å Release Date: 2013-02-06 Classification: transferase/transferase inhibitor Ligands: IPA, 1BR |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-02-06
Ligands: IPA, 1BR
![]() |
Structure Of Focal Adhesion Kinase Catalytic Domain In Complex With Novel Allosteric Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.67 Å Release Date: 2012-08-22 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 0O7, IPA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-08-22
Ligands: 0O7, IPA
![]() |
Structure Of Focal Adhesion Kinase Catalytic Domain In Complex With Novel Allosteric Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.65 Å Release Date: 2012-07-25 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 0PF |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-07-25
Ligands: 0PF
