Search Count: 75
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Crystal Structures Of Apo Keap1, Keap1-Peptide, And Keap1-Compound Complexes
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2014-08-20 Classification: TRANSCRIPTION |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-08-20
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Selective & Brain-Permeable Polo-Like Kinase-2 (Plk-2) Inhibitors That Reduce -Synuclein Phosphorylation In Rat Brain
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2013-12-25 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: R78 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-12-25
Ligands: R78
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Selective & Brain-Permeable Polo-Like Kinase-2 (Plk-2) Inhibitors That Reduce -Synuclein Phosphorylation In Rat Brain
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.74 Å Release Date: 2013-12-25 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 1D1 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-12-25
Ligands: 1D1
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Crystal Structures Of Apo Keap1, Keap1-Peptide, And Keap1-Compound Complexes
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2013-12-18 Classification: TRANSCRIPTION |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-12-18
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Crystal Structures Of Apo Keap1, Keap1-Peptide, And Keap1-Compound Complexes
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2013-12-18 Classification: TRANSCRIPTION Ligands: 12O |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-12-18
Ligands: 12O
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Selective & Brain-Permeable Polo-Like Kinase-2 (Plk-2) Inhibitors That Reduce -Synuclein Phosphorylation In Rat Brain
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2013-11-20 Classification: transferase/transferase inhibitor Ligands: 11G |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-11-20
Ligands: 11G
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Selective & Brain-Permeable Polo-Like Kinase-2 (Plk-2) Inhibitors That Reduce -Synuclein Phosphorylation In Rat Brain
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.90 Å Release Date: 2013-11-20 Classification: transferase/transferase inhibitor Ligands: 1C7 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-11-20
Ligands: 1C7
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Design And Synthesis Of Thiophene Dihydroisoquinolins As Novel Bace-1 Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.91 Å Release Date: 2013-10-09 Classification: hydrolase/hydrolase inhibitor Ligands: ZN, 1B7 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-10-09
Ligands: ZN, 1B7
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Selective & Brain-Permeable Polo-Like Kinase-2 (Plk-2) Inhibitors That Reduce Alpha-Synuclein Phosphorylation In Rat Brain
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.91 Å Release Date: 2013-08-14 Classification: transferase/transferase inhibitor Ligands: 1C8 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-08-14
Ligands: 1C8
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Structure Of Parkin-S223P E3 Ligase
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.58 Å Release Date: 2013-06-19 Classification: LIGASE Ligands: ZN, BA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-06-19
Ligands: ZN, BA
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Structure Of Parkin E3 Ligase
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2013-06-19 Classification: LIGASE Ligands: ZN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-06-19
Ligands: ZN
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Design And Synthesis Of Brain Penetrant Selective Jnk Inhibitors With Improved Pharmacokinetic Properties For The Prevention Of Neurodegeneration
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2013-05-08 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 34I |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-05-08
Ligands: 34I
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Crystal Structure Of Kit Kinase Domain With A Small Molecule Inhibitor, Plx647
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2013-03-27 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 647 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-03-27
Ligands: 647
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Crystal Structure Of Fms Kinase Domain With A Small Molecular Inhibitor, Plx647-Ome
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.90 Å Release Date: 2013-03-27 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 64M |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-03-27
Ligands: 64M
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Structure-Based Design Of Novel Dihydroisoquinoline Bace-1 Inhibitors That Do Not Engage The Catalytic Aspartates
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2013-03-06 Classification: hydrolase/hydrolase inhibitor Ligands: ZN, 0ZA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-03-06
Ligands: ZN, 0ZA
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Design And Synthesis Of Thiophene Dihydroisoquinolins As Novel Bace-1 Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2013-03-06 Classification: hydrolase/hydrolase inhibitor Ligands: ZN, 1B8 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-03-06
Ligands: ZN, 1B8
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Design And Synthesis Of Thiophene Dihydroisoquinolins As Novel Bace-1 Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2013-03-06 Classification: hydrolase/hydrolase inhibitor Ligands: ZN, 1BF |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-03-06
Ligands: ZN, 1BF
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Design And Synthesis Of Thiophene Dihydroisoquinolins As Novel Bace-1 Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.78 Å Release Date: 2013-03-06 Classification: hydrolase/hydrolase inhibitor Ligands: ZN, 1B9 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-03-06
Ligands: ZN, 1B9
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Structure-Based Design Of Novel Dihydroisoquinoline Bace-1 Inhibitors That Do Not Engage The Catalytic Aspartates
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2013-03-06 Classification: hydrolase/hydrolase inhibitor Ligands: 1BB, ZN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-03-06
Ligands: 1BB, ZN
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Structure-Based Design Of Novel Dihydroisoquinoline Bace-1 Inhibitors That Do Not Engage The Catalytic Aspartates
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.07 Å Release Date: 2013-03-06 Classification: hydrolase/hydrolase inhibitor Ligands: ZN, 1BS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-03-06
Ligands: ZN, 1BS