Search Count: 23
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Salt-Inducible Kinase 3 In Complex With An Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.10 Å Release Date: 2024-01-10 Classification: SIGNALING PROTEIN Ligands: VRU |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-01-10
Ligands: VRU
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Il-17A In Complex With Small Molecule Modulators
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.48 Å Release Date: 2022-04-20 Classification: IMMUNE SYSTEM Ligands: RMK |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-04-20
Ligands: RMK
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Il-17A In Complex With Small Molecule Modulators
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.18 Å Release Date: 2022-04-20 Classification: IMMUNE SYSTEM Ligands: RMQ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-04-20
Ligands: RMQ
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Crystal Structure Of The Rbpj-Notch1-Nrarp Ternary Complex Bound To Dna
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.75 Å Release Date: 2019-08-14 Classification: DNA BINDING PROTEIN/DNA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-08-14
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Crystal Structure Of Trk-A In Complex With The Pan-Trk Kinase Inhibitor, Compound 10B.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.68 Å Release Date: 2018-07-11 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: FKY |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-07-11
Ligands: FKY
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Crystal Structure Of Trk-A In Complex With The Pan-Trk Kinase Inhibitor, Compound 13B.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.53 Å Release Date: 2018-07-11 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 22L, GO7 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-07-11
Ligands: 22L, GO7
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Crystal Structure Of Trk-A In Complex With The Pan-Trk Kinase Inhibitor, Compound 19.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.11 Å Release Date: 2018-07-11 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 22L, GOD |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-07-11
Ligands: 22L, GOD
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Crystal Structure Of Trk-A In Complex With The Pan-Trk Kinase Inhibitor, Compound 3.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.91 Å Release Date: 2018-07-11 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: GXA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-07-11
Ligands: GXA
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Crystal Structure Of Trka In Complex With Pf-00593174
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.07 Å Release Date: 2017-03-01 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: 6K0 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-03-01
Ligands: 6K0
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Crystal Structure Of Trka In Complex With Pf-05206283
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.59 Å Release Date: 2017-03-01 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: 6K1 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-03-01
Ligands: 6K1
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Crystal Structure Of Trka In Complex With Pf-05247452
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.52 Å Release Date: 2017-03-01 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: 6K2 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-03-01
Ligands: 6K2
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Crystal Structure Of Trka In Complex With Pf-06273340
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.63 Å Release Date: 2017-03-01 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: 6K4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-03-01
Ligands: 6K4
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Inhibition Of Small Gtpases By Stabilization Of The Gdp Complex, A Novel Approach Applied To Rit1, A Target For Rheumatoid Arthritis
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2014-09-17 Classification: PROTEIN BINDING Ligands: GDP, MG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-09-17
Ligands: GDP, MG
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Truncation And Optimisation Of Peptide Inhibitors Of Cdk2, Cyclin A Through Structure Guided Design
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2009-06-09 Classification: TRANSFERASE Ligands: CK7 |
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION
Release Date: 2009-06-09
Ligands: CK7
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Truncation And Optimisation Of Peptide Inhibitors Of Cdk2, Cyclin A Through Structure Guided Design
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION Resolution:2.53 Å Release Date: 2009-06-09 Classification: TRANSFERASE |
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION
Release Date: 2009-06-09
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Truncation And Optimisation Of Peptide Inhibitors Of Cdk2, Cyclin A Through Structure Guided Design
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION Resolution:2.90 Å Release Date: 2009-06-09 Classification: TRANSFERASE |
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION
Release Date: 2009-06-09
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Replace: A Strategy For Iterative Design Of Cyclin Binding Groove Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2008-01-29 Classification: TRANSFERASE Ligands: C35 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-01-29
Ligands: C35
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Replace: A Strategy For Iterative Design Of Cyclin Binding Groove Inhibitors
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION Resolution:2.06 Å Release Date: 2007-03-27 Classification: TRANSFERASE/INHIBITOR Ligands: MTZ, GVC |
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION
Release Date: 2007-03-27
Ligands: MTZ, GVC
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Cyclin A Binding Groove Inhibitor H-Arg-Arg-Leu-Ile-Phe-Nh2
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2003-12-11 Classification: TRANSFERASE/TRANSFERASE INHIBITOR |
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION
Release Date: 2003-12-11
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Cyclin A Binding Groove Inhibitor Ac-Arg-Arg-Leu-Asn-(M-Cl-Phe)-Nh2
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2003-12-11 Classification: TRANSFERASE/TRANSFERASE INHIBITOR |
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION
Release Date: 2003-12-11
