Search Count: 7
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Crystal Structure Of Beta-Site App-Cleaving Enzyme 1 Complexed With N-(3-((4As,7As)-2-Amino-4,4A,5,6-Tetrahydro-7Ah-Furo[2,3-D][1,3]Thiazin-7A-Yl)-4-Fluorophenyl)-5-Bromo-2-Pyridinecarboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.51 Å Release Date: 2016-11-23 Classification: HYDROLASE Ligands: 7H3 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-11-23
Ligands: 7H3
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Compound 10
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.98 Å Release Date: 2016-10-05 Classification: Hydrolase/Hydrolase Inhibitor Ligands: GOL, IOD, 5QU |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-10-05
Ligands: GOL, IOD, 5QU
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(4~{S},6~{S})-4-[2,4-Bis(Fluoranyl)Phenyl]-4-Methyl-6-Pyrimidin-5-Yl-5,6-Dihydro-1,3-Thiazin-2-Amine (Compound 12) Bound To Bace1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.98 Å Release Date: 2016-09-07 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: 6WD |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-09-07
Ligands: 6WD
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(4~{S},6~{S})-4-[2,4-Bis(Fluoranyl)Phenyl]-6-(3,5-Dimethyl-1,2-Oxazol-4-Yl)-4-Methyl-5,6-Dihydro-1,3-Thiazin-2-Amine (Compound 5) Bound To Bace1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.12 Å Release Date: 2016-09-07 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: IOD, 6WE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-09-07
Ligands: IOD, 6WE
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Compound 18
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.11 Å Release Date: 2016-07-06 Classification: Hydrolase/Hydrolase Inhibitor Ligands: GOL, IOD, 5QV |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-07-06
Ligands: GOL, IOD, 5QV
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Novel Cdk-5 Inhibitors - Crystal Structure Of Inhibitor Efp With Cdk-2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2009-09-08 Classification: TRANSFERASE Ligands: EFP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2009-09-08
Ligands: EFP
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Novel Cdk-5 Inhibitors - Crystal Structure Of Inhibitor Efq With Cdk-2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2009-09-08 Classification: TRANSFERASE Ligands: EFQ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2009-09-08
Ligands: EFQ
