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A New Class Of Hiv-1 Protease Inhibitor: The Crystallographic Structure, Inhibition And Chemical Synthesis Of An Aminimide Peptide Isostere
Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 1997-09-17 Classification: ASPARTYL PROTEASE Ligands: ARQ |
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Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 1997-08-20 Classification: ASPARTYL PROTEASE Ligands: NMB |
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Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 1997-09-17 Classification: ASPARTYL PROTEASE Ligands: AH1 |
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Structure Of A Non-Peptide Inhibitor Complexed With Hiv-1 Protease: Developing A Cycle Of Structure-Based Drug Design
Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 1997-10-15 Classification: ASPARTYL PROTEASE Ligands: CL, THK |
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Active-Site Mobility In Human Immunodeficiency Virus Type 1 Protease As Demonstrated By Crystal Structure Of A28S Mutant
Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 1998-04-15 Classification: ASPARTYL PROTEASE Ligands: U0E |
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Organism: Simian immunodeficiency virus
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 1998-05-27 Classification: ASPARTYL PROTEASE |
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Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 1998-04-15 Classification: ASPARTYL PROTEASE Ligands: DMQ |
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Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 1998-04-15 Classification: ASPARTYL PROTEASE Ligands: DMP |
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Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 1998-04-15 Classification: ASPARTYL PROTEASE Ligands: DMP |
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Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 1999-03-23 Classification: ASPARTYL PROTEASE Ligands: 216 |
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Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 1997-10-15 Classification: ASPARTYL PROTEASE Ligands: 846 |
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Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 1998-04-15 Classification: ASPARTYL PROTEASE Ligands: DMP |
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Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 1997-10-15 Classification: ASPARTYL PROTEASE Ligands: 146 |
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Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 1997-10-15 Classification: ASPARTYL PROTEASE Ligands: DMP |
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Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 1997-10-15 Classification: ASPARTYL PROTEASE Ligands: XV6 |
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G48H Mutant Of Hiv-1 Protease In Complex With A Peptidic Inhibitor U-89360E
Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 1998-06-17 Classification: ASPARTYL PROTEASE Ligands: U0E |
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Organism: Human immunodeficiency virus 1
Method: SOLUTION NMR Release Date: 1996-08-17 Classification: ASPARTYL PROTEASE Ligands: DMP |
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Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 1998-12-09 Classification: ASPARTYL PROTEASE Ligands: BAY |
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Organism: Human immunodeficiency virus 1
Method: SOLUTION NMR Release Date: 1996-08-17 Classification: ASPARTYL PROTEASE Ligands: DMP |
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Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 1999-01-13 Classification: ASPARTYL PROTEASE Ligands: BAY |




















